The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 2.8M data for 1.2M Compounds and 9.2K Targets. Of those, 1,346K data for 622K Compounds and 4.5K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

Advanced Search

17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities.EBI
University Of Paris
Investigation of subsite preferences in aminopeptidase A (EC 3.4.11.7) led to the design of the first highly potent and selective inhibitors of this enzyme.EBI
University Of Paris
Optimal recognition of neutral endopeptidase and angiotensin-converting enzyme active sites by mercaptoacyldipeptides as a means to design potent dual inhibitors.EBI
University Of Paris
Design of orally active dual inhibitors of neutral endopeptidase and angiotensin-converting enzyme with long duration of action.EBI
University Of Paris
Hydroxamic acids as potent inhibitors of endothelin-converting enzyme from human bronchiolar smooth muscle.EBI
Berlex Laboratories
New thiol inhibitors of neutral endopeptidase EC 3.4.24.11: synthesis and enzyme active-site recognition.EBI
University Of Paris
Enkephalinase inhibitors. 1. 2,4-Dibenzylglutaric acid derivatives.EBI
Ciba-Geigy
Retro-inverso concept applied to the complete inhibitors of enkephalin-degrading enzymes.EBI
Ua 498 Cnrs
 
Kelatorphan and related analogs: potent and selective inhibitors of leukotriene A4 hydrolaseEBI
TBA
Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder.EBI
Pfizer
Novel selective inhibitors of neutral endopeptidase for the treatment of female sexual arousal disorder. Synthesis and activity of functionalized glutaramides.EBI
Pfizer
N-[2-(Indan-1-yl)-3-mercapto-propionyl] amino acids as highly potent inhibitors of the three vasopeptidases (NEP, ACE, ECE): In vitro and In vivo activities.EBI
University Of Paris
Exploration of neutral endopeptidase active site by a series of new thiol-containing inhibitors.EBI
University Of Paris
Mercaptoacyl amino acid inhibitors of atriopeptidase. 1. Structure-activity relationship studies of methionine and S-alkylcysteine derivatives.EBI
Schering-Plough Research Institute
New kelatorphan-related inhibitors of enkephalin metabolism: improved antinociceptive properties.EBI
University Of Paris
Carboxyalkyl dipeptides with atrial natriuretic factor potentiating and antihypertensive activity.EBI
Schering-Plough Research Institute