17 articles for PK Jadhav
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Discovery of Cathepsin S Inhibitor LY3000328 for the Treatment of Abdominal Aortic Aneurysm.

Eli Lilly
Synthesis of 7-membered cyclic hydroxyguanidines: Novel HIV-1 protease inhibitors

TBA
(S)-N-{3-[1-cyclopropyl-1-(2,4-difluoro-phenyl)-ethyl]-1H-indol-7-yl}-methanesulfonamide: a potent, nonsteroidal, functional antagonist of the mineralocorticoid receptor.

Eli Lilly
Synthesis and biological evaluation of nonpeptide integrin antagonists containing spirocyclic scaffolds.

Pharmaceutical Research Institute
Disubstituted indazoles as potent antagonists of the integrin alpha(v)beta(3).

Dupont Pharmaceuticals
Isoxazolines as potent antagonists of the integrin alpha(v)beta(3).

Dupont Pharmaceuticals
Rapid synthesis of RGD mimetics with isoxazoline scaffolds on solid phase: identification of alphavbeta3 antagonists lead compounds.

Dupont Pharmaceuticals
Cyclic HIV protease inhibitors: design and synthesis of orally bioavailable, pyrazole P2/P2' cyclic ureas with improved potency.

Dupont Pharmaceuticals
Cyclic urea amides: HIV-1 protease inhibitors with low nanomolar potency against both wild type and protease inhibitor resistant mutants of HIV.

Dupont Pharmaceuticals
Pyrrolidine amide compounds as histone demethylase inhibitors

Genentech
Compositions, methods, and systems for the synthesis and use of imaging agents

Lantheus Medical Imaging
PRMT5 inhibitors and uses thereof

Epizyme
Structure-activity relationship of HIV-1 protease inhibitors containing AHPBA. Part III: Modification of P2 site.

Sankyo
Structure-activity relationships of HIV-1 PR inhibitors containing AHPBA--II. Modification of pyrrolidine ring at P1' proline.

Sankyo
5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.

Merck Research Laboratories
Aminodiol HIV protease inhibitors. Synthesis and structure-activity relationships of P1/P1' compounds: correlation between lipophilicity and cytotoxicity.

Bristol-Myers Squibb
Synthesis and structure-activity relationships of a series of penicillin-derived HIV proteinase inhibitors containing a stereochemically unique peptide isostere.

Glaxo Group Research