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21 articles for T Noguchi-Yachide


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of N-(1-(3-(4-phenoxyphenyl)-1,2,4-oxadiazol-5-yl)ethyl)acetamides as novel acetyl-CoA carboxylase 2 (ACC2) inhibitors with peroxisome proliferator-activated receptora/d (PPARa/d) dual agonistic activity.EBI
The University of Tokyo
Effects of alkyl side chains and terminal hydrophilicity on vitamin D receptor (VDR) agonistic activity based on the diphenylpentane skeleton.EBI
National Institute of Health Sciences
Discovery and structure-activity relationship studies of N6-benzoyladenine derivatives as novel BRD4 inhibitors.EBI
The University of Tokyo
Structure-activity relationships of oxysterol-derived pharmacological chaperones for Niemann-Pick type C1 protein.EBI
The University of Tokyo
Structure-activity relationship of benzodiazepine derivatives as LXXLL peptide mimetics that inhibit the interaction of vitamin D receptor with coactivators.EBI
The University of Tokyo
Small-molecular, non-peptide, non-ATP-competitive polo-like kinase 1 (Plk1) inhibitors with a terphenyl skeleton.EBI
The University of Tokyo
Design, synthesis, and biological evaluation of novel transrepression-selective liver X receptor (LXR) ligands with 5,11-dihydro-5-methyl-11-methylene-6H-dibenz[b,e]azepin-6-one skeleton.EBI
The University of Tokyo
Novel selective anti-androgens with a diphenylpentane skeleton.EBI
The University of Tokyo
LXXLL peptide mimetics as inhibitors of the interaction of vitamin D receptor with coactivators.EBI
The University of Tokyo
beta-Naphthoflavone analogs as potent and soluble aryl hydrocarbon receptor agonists: improvement of solubility by disruption of molecular planarity.EBI
The University of Tokyo
Separation of alpha-glucosidase-inhibitory and liver X receptor-antagonistic activities of phenethylphenyl phthalimide analogs and generation of LXRalpha-selective antagonists.EBI
The University of Tokyo
Liver X receptor antagonists with a phthalimide skeleton derived from thalidomide-related glucosidase inhibitors.EBI
University of Tokyo
Physicochemical characterization of EBI
Tokyo Medical and Dental University
Design, synthesis and structure-activity relationship of 4-(1,1,1,3,3,3-hexafluoro-2-hydroxyisoprop-2-yl)phenylsilane derivatives as liver X receptor agonists.EBI
Tokyo Medical and Dental University
Structure-activity relationship studies of non-carboxylic acid peroxisome proliferator-activated receptor α/δ (PPARα/δ) dual agonists.EBI
The University of Tokyo
Structure-activity relationship study of estrogen receptor down-regulators with a diphenylmethane skeleton.EBI
The University of Tokyo
Phenanthridin-6-one derivatives as the first class of non-steroidal pharmacological chaperones for Niemann-Pick disease type C1 protein.EBI
The University of Tokyo
Design and synthesis of estrogen receptor ligands with a 4-heterocycle-4-phenylheptane skeleton.EBI
Nagasaki University
Synthesis and evaluation of novel dual BRD4/HDAC inhibitors.EBI
The University of Tokyo
Switching subtype-selectivity: Fragment replacement strategy affords novel class of peroxisome proliferator-activated receptorα/δ (PPARα/δ) dual agonists.EBI
The University of Tokyo
Therapeutic compounds and uses thereofBDB
Genentech