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13 articles for AM Kral


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
8
Delayed and Prolonged Histone Hyperacetylation with a Selective HDAC1/HDAC2 Inhibitor.EBI
Merck Research Laboratories
63
Exploration of the internal cavity of histone deacetylase (HDAC) with selective HDAC1/HDAC2 inhibitors (SHI-1:2).EBI
Merck Research Laboratories
2
Phenylglycine and phenylalanine derivatives as potent and selective HDAC1 inhibitors (SHI-1).EBI
Merck Research Laboratories
19
Rapid assembly of diverse and potent allosteric Akt inhibitors.EBI
Merck Research Laboratories
22
Exploring the pharmacokinetic properties of phosphorus-containing selective HDAC 1 and 2 inhibitors (SHI-1:2).EBI
Merck Research Laboratories
39
SAR profiles of spirocyclic nicotinamide derived selective HDAC1/HDAC2 inhibitors (SHI-1:2).EBI
Merck Research Laboratories
19
Optimization of biaryl Selective HDAC1&2 Inhibitors (SHI-1:2).EBI
Merck Research Laboratories
42
The discovery of 6-amino nicotinamides as potent and selective histone deacetylase inhibitors.EBI
Merck Research Laboratories
22
Design of novel histone deacetylase inhibitors.EBI
Merck Research Laboratories
7
2-substituted piperazines as constrained amino acids. Application to the synthesis of potent, non carboxylic acid inhibitors of farnesyltransferase.EBI
Merck Research Laboratories
18
Aminoindazole derivatives as sodium channel inhibitorsBDB
Almirall
116
P2X7 modulatorsBDB
Janssen Pharmaceutica
30
Structure-activity relationships of a new family of steroidal aromatase inhibitors. 1. Synthesis and evaluation of a series of analogs related to 19-[(methylthio)methyl]androstenedione (RU54115).BDB
Centre De Recherche De Roussel Uclaf