34 articles for PJ Scammells
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Synthesis, Biological Evaluation, and Utility of Fluorescent Ligands Targeting theµ-Opioid Receptor.
University of Nottingham
Synthesis and pharmacological evaluation of dual acting ligands targeting the adenosine A2A and dopamine D2 receptors for the potential treatment of Parkinson's disease.
Monash University (Parkville Campus)
Ligand-induced conformational change of Plasmodium falciparum AMA1 detected using 19F NMR.
La Trobe University
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M1 muscarinic acetylcholine receptor.
Monash University (Parkville Campus)
A structure-activity analysis of biased agonism at the dopamine D2 receptor.
Monash University (Parkville Campus)
Synthesis and pharmacological evaluation of dual acting antioxidant A(2A) adenosine receptor agonists.
Monash University
N6-substituted C5'-modified adenosines as A1 adenosine receptor agonists.
Monash University (Parkville Campus)
Structure-activity relationships of adenosines with heterocyclic N6-substituents.
Monash University (Parkville Campus)
Structure-based optimization and biological evaluation of human 20a-hydroxysteroid dehydrogenase (AKR1C1) salicylic acid-based inhibitors.
Monash University (Parkville Campus)
Synthesis and evaluation of new N6-substituted adenosine-5'-N-methylcarboxamides as A3 adenosine receptor agonists.
Monash University
3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonists.
Monash University (Parkville Campus)
Structure-guided design, synthesis, and evaluation of salicylic acid-based inhibitors targeting a selectivity pocket in the active site of human 20alpha-hydroxysteroid dehydrogenase (AKR1C1).
Monash University (Parkville Campus)
2-aminothienopyridazines as novel adenosine A1 receptor allosteric modulators and antagonists.
Monash University
Dual acting antioxidant A1 adenosine receptor agonists.
Monash University (Parkville Campus)
The Design, Synthesis, and Evaluation of Novel 9-Arylxanthenedione-Based Allosteric Modulators for the δ
Monash University (Parkville Campus)
Development and Application of Subtype-Selective Fluorescent Antagonists for the Study of the Human Adenosine A
Monash University
2-Amino-3-benzoylthiophene allosteric enhancers of A1 adenosine agonist binding: new 3, 4-, and 5-modifications.
Deakin University
New irreversible adenosine A(1) antagonists based on FSCPX.
Monash University (Parkville Campus)
Rapid Elaboration of Fragments into Leads by X-ray Crystallographic Screening of Parallel Chemical Libraries (REFiL
Monash University (Parkville Campus)
Fluorosulfonyl-substituted xanthines as selective irreversible antagonists for the A(1)-adenosine receptor.
Deakin University
Structure-Kinetic Profiling of Haloperidol Analogues at the Human Dopamine D
University of Nottingham
Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions.
Monash University
Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases.
Monash University
Two-pronged attack: dual inhibition of Plasmodium falciparum M1 and M17 metalloaminopeptidases by a novel series of hydroxamic acid-based inhibitors.
Monash University
Substituted 1,3-dipropylxanthines as irreversible antagonists of A1 adenosine receptors.
University of South Florida
Synthesis and pharmacological profiling of analogues of benzyl quinolone carboxylic acid (BQCA) as allosteric modulators of the M1 muscarinic receptor.
Monash University
Novel adenosine A(2A) receptor ligands: a synthetic, functional and computational investigation of selected literature adenosine A(2A) receptor antagonists for extending into extracellular space.
Monash University (Parkville Campus)
Synthesis and Pharmacological Evaluation of Heterocyclic Carboxamides: Positive Allosteric Modulators of the M
Monash University (Parkville Campus)
Synthesis and adenosine receptor affinity of a series of pyrazolo[3,4-d]pyrimidine analogues of 1-methylisoguanosine.
Griffith University
