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23 articles for AD Mesecar


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
8
Probing the structural requirements of non-electrophilic naphthalene-based Nrf2 activators.EBI
University of Illinois At Chicago
15
Structure-based design, synthesis and biological evaluation of novelß-secretase inhibitors containing a pyrazole or thiazole moiety as the P3 ligand.EBI
Purdue University
7
X-ray structural and biological evaluation of a series of potent and highly selective inhibitors of human coronavirus papain-like proteases.EBI
Purdue University
10
Synthesis of 3-(3-aryl-pyrrolidin-1-yl)-5-aryl-1,2,4-triazines that have antibacterial activity and also inhibit inorganic pyrophosphatase.EBI
Purdue University
35
Design, synthesis, biological and structural evaluation of functionalized resveratrol analogues as inhibitors of quinone reductase 2.EBI
Purdue University
5
Synthesis of novel¿¿3 receptor ligands via an unusual Knoevenagel condensation.EBI
Moscow State University
26
Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancer.EBI
Purdue University
28
Design and synthesis of 2-pyridones as novel inhibitors of the Bacillus anthracis enoyl-ACP reductase.EBI
University of Illinois At Chicago
17
Design, synthesis, and biological evaluation of potent quinoline and pyrroloquinoline ammosamide analogues as inhibitors of quinone reductase 2.EBI
Purdue University
25
Potential chemopreventive agents based on the structure of the lead compound 2-bromo-1-hydroxyphenazine, isolated from Streptomyces species, strain CNS284.EBI
Purdue University
6
Bioactive compounds from the fern Lepisorus contortus.EBI
Yunnan Normal University
16
Exploration of P1 and P4 modifications of nirmatrelvir: Design, synthesis, biological evaluation, and X-ray structural studies of SARS-CoV-2 Mpro inhibitors.EBI
Purdue University
20
SARS-CoV-2 papain-like protease (PLpro) inhibitory and antiviral activity of small molecule derivatives for drug leads.EBI
Purdue University
2
Design and synthesis of peptidomimetic severe acute respiratory syndrome chymotrypsin-like protease inhibitors.EBI
Purdue University
7
Structure-based design, synthesis, and biological evaluation of peptidomimetic SARS-CoV 3CLpro inhibitors.EBI
Purdue University
10
Design, synthesis, X-ray studies, and biological evaluation of novel BACE1 inhibitors with bicyclic isoxazoline carboxamides as the P3 ligand.EBI
Purdue University
17
Design, synthesis, and X-ray structural studies of BACE-1 inhibitors containing substituted 2-oxopiperazines as P1'-P2' ligands.EBI
Purdue University
37
Pyrazole compounds substituted with heteroaryl and pharmaceutical use thereofBDB
Japan Tobacco
124
Pyrazolopyridinamines as MKNK1 and MKNK2 inhibitorsBDB
Bayer
80
Ectonucleotidase inhibitors and methods of use thereofBDB
Calithera Biosciences
8
Metabolism probes for therapy and diagnosisBDB
Vanderbilt University
14
Oxathiolane carboxylic acids and derivatives for the treatment and prophylaxis of virus infectionBDB
Hoffmann-La Roche
16
Diprolyl nitriles as potent dipeptidyl peptidase IV inhibitors.BDB
Bristol Myers Squibb