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14 articles for JA Markwalder


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification and optimization of a novel series of indoleamine 2,3-dioxygenase inhibitors.EBI
Bristol-Myers Squibb Research and Development
Synthesis and biological activities of potential metabolites of the non-nucleoside reverse transcriptase inhibitor efavirenz.EBI
Dupont Pharmaceuticals
3,3a-Dihydropyrano[4,3,2-de]quinazolin-2(1H)-ones are potent non-nucleoside reverse transcriptase inhibitors.EBI
Dupont Pharmaceuticals
Synthesis and biological evaluation of biaryl alkyl ethers as inhibitors of IDO1.EBI
Bristol Myers Squibb
Development of a series of novel o-phenylenediamine-based indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors.EBI
Bristol-Myers Squibb Research and Development
Modified biotin, mutant streptavidin, and use thereofBDB
Savid Therapeutics
Oxysterol-binding protein (OSBP)-related protein 4 (ORP4) is essential for cell proliferation and survival.BDB
Dalhousie University
Substituted imidazopyrazines as Akt kinase inhibitorsBDB
Bayer Pharma Aktiengesellschaft
Rapid Evolution of 6-Phenylpurine Inhibitors of Protein Kinase B through Structure-Based Design.BDB
Astex
5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.BDB
Merck Research Laboratories
Multidrug resistance to HIV-1 protease inhibition requires cooperative coupling between distal mutations.BDB
The Johns Hopkins University
Identification of potent and selective small-molecule inhibitors of caspase-3 through the use of extended tethering and structure-based drug design.BDB
Sunesis Pharmaceuticals
Aza-peptide analogs as potent human immunodeficiency virus type-1 protease inhibitors with oral bioavailability.BDB
Ciba-Geigy