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19 articles for LF Hennequin


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of novel TACE inhibitors compatible with topical application.EBI
Nestl�
Discovery of phenoxyindazoles and phenylthioindazoles as ROR¿ inverse agonists.EBI
Galderma R & D
Discovery of AZD8931, an Equipotent, Reversible Inhibitor of Signaling by EGFR, HER2, and HER3 Receptors.EBI
Astrazeneca
Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase.EBI
Astrazeneca
Inhibitors of epidermal growth factor receptor tyrosine kinase: optimisation of potency and in vivo pharmacokinetics.EBI
Astrazeneca
Novel 4-anilinoquinazolines with C-6 carbon-linked side chains: synthesis and structure-activity relationship of a series of potent, orally active, EGF receptor tyrosine kinase inhibitors.EBI
Astrazeneca
Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket.EBI
Astrazeneca
5-Substituted 4-anilinoquinazolines as potent, selective and orally active inhibitors of erbB2 receptor tyrosine kinase.EBI
Astrazeneca
Impact of Minor Structural Modifications on Properties of a Series of mTOR Inhibitors.EBI
Nestl�
Design and synthesis of potent non-polyglutamatable quinazoline antifolate thymidylate synthase inhibitors.EBI
Astrazeneca
Quinazoline antifolates thymidylate synthase inhibitors: lipophilic analogues with modification to the C2-methyl substituent.EBI
Zeneca Pharma
Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma.EBI
Nestle Skin Health R&D
Sulfoximines as potent RORγ inverse agonists.EBI
Nestle Skin Health
Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis.EBI
Nestle Skin Health
Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne.EBI
Nestl�
Azapeptides as CD36 binding compoundsBDB
Valorisation-Recherche, Limited Partnership
Selective octahydro-cyclopenta[C] pyrrole negative modulators of NR2BBDB
Cadent Therapeutics
C17-aryl substituted betulinic acid analogsBDB
Viiv Healthcare UK (NO.5)
Tyrosine kinase inhibitors. 1. Structure-activity relationships for inhibition of epidermal growth factor receptor tyrosine kinase activity by 2,3-dihydro-2-thioxo-1H-indole-3-alkanoic acids and 2,2'-dithiobis(1H-indole-3-alkanoic acids).BDB
University of Auckland