18 articles for DA Erlanson
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Fragment-to-Lead Medicinal Chemistry Publications in 2015.

Astex Pharmaceuticals
Fragment-based drug discovery.

Sunesis Pharmaceuticals
Discovery of an Aurora kinase inhibitor through site-specific dynamic combinatorial chemistry.

Sunesis Pharmaceuticals
Fragment-to-Lead Medicinal Chemistry Publications in 2022.

Astex Pharmaceuticals
Fragment-to-Lead Medicinal Chemistry Publications in 2021.

Astex Pharmaceuticals
Fragment-to-Lead Medicinal Chemistry Publications in 2020.

Vrije Universiteit Amsterdam
Utilizing structure based drug design and metabolic soft spot identification to optimize the in vitro potency and in vivo pharmacokinetic properties leading to the discovery of novel reversible Bruton's tyrosine kinase inhibitors.

Biogen
Fragment-to-Lead Medicinal Chemistry Publications in 2019.

Novartis Institutes For Biomedical Research
Fragment-to-Lead Medicinal Chemistry Publications in 2017.

Astex Pharmaceuticals
Optimization of novel reversible Bruton's tyrosine kinase inhibitors identified using Tethering-fragment-based screens.

Biogen
Fragment-to-Lead Medicinal Chemistry Publications in 2018.

Frontier Medicines
Discovery of

Amgen
Fragment-to-Lead Medicinal Chemistry Publications in 2016.

Astex Pharmaceuticals
Small molecule inhibitors of GPCR GPR68 and related receptors for treating cancer, glioblastoma, and other indications

University of Maryland, Baltimore
4-oxo-3,4-dihydro-1,2,3-benzotriazine modulators of GPR139

Takeda Pharmaceutical
Quinazoline-urea, new protein kinase inhibitors in treatment of prostate cancer.

Universit�� Lille Nord De France
Design, synthesis, and anticonvulsant activity of some derivatives of xanthone with aminoalkanol moieties.

Jagiellonian University Medical College
Methods of treating retroviral infections and related dosage regimes

Chimerix