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20 articles for A Bedini


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.EBI
University of Urbino
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties.EBI
University of Urbino
Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: synthesis, binding affinity and intrinsic activity for MT(1) and MT(2) melatonin receptors.EBI
University of Urbino
Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminus.EBI
University of Bologna
Antiangiogenic effect of dual/selective alpha(5)beta(1)/alpha(v)beta(3) integrin antagonists designed on partially modified retro-inverso cyclotetrapeptide mimetics.EBI
Universita Degli Studi Di Bologna
Diphenidol-related diamines as novel muscarinic M4 receptor antagonists.EBI
University of Bologna
Synthesis and biological activity of new melatonin dimeric derivatives.EBI
Università
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MTEBI
University of Urbino Carlo Bo
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma.EBI
University of Parma
Versatile Picklocks To Access All Opioid Receptors: Tuning the Selectivity and Functional Profile of the Cyclotetrapeptide c[Phe-d-Pro-Phe-Trp] (CJ-15,208).EBI
University of Bologna
(E)-3-(2-(N-phenylcarbamoyl)vinyl)pyrrole-2-carboxylic acid derivatives. A novel class of glycine site antagonists.EBI
Università
Synthesis of tripeptides containing D-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception.EBI
University of Bologna
N-(substituted-anilinoethyl)amides: design, synthesis, and pharmacological characterization of a new class of melatonin receptor ligands.EBI
University of Parma
Analysis of structure-activity relationships for MT2 selective antagonists by melatonin MT1 and MT2 receptor models.EBI
University of Parma
Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity.EBI
University of Milan
Three-dimensional quantitative structure-activity relationship studies on selected MT1 and MT2 melatonin receptor ligands: requirements for subtype selectivity and intrinsic activity modulation.EBI
University of Parma
Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit.EBI
University of Urbino
Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist.EBI
University of Bologna
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands.EBI
University of Parma
Structural basis for binding and selectivity of antimalarial and anticancer ethylenediamine inhibitors to protein farnesyltransferase.BDB
Duke University Medical Center