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28 articles for A Saeed


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Quinazolines and quinazolinones as ubiquitous structural fragments in medicinal chemistry: An update on the development of synthetic methods and pharmacological diversification.EBI
Quaid-I-Azam University
Isocoumarins, miraculous natural products blessed with diverse pharmacological activities.EBI
Quaid-I-Azam University
2-Chloro-4-[[(1R,2R)-2-hydroxy-2-methyl-cyclopentyl]amino]-3-methyl-benzonitrile: A Transdermal Selective Androgen Receptor Modulator (SARM) for Muscle Atrophy.EBI
Eli Lilly
Synthetic approaches, functionalization and therapeutic potential of quinazoline and quinazolinone skeletons: the advances continue.EBI
University of Nottingham
Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: synthetic approaches and multifarious applications.EBI
Quaid-I-Azam University
New aminobenzenesulfonamide-thiourea conjugates: synthesis and carbonic anhydrase inhibition and docking studies.EBI
Comsats Institute of Information Technology
Synthesis, cytotoxicity and molecular modelling studies of new phenylcinnamide derivatives as potent inhibitors of cholinesterases.EBI
Quaid-I-Azam University
Identification of sulfonic acids as efficient ecto-5'-nucleotidase inhibitors.EBI
Comsats Institute of Information Technology
3-Amino-5,5-dimethylhexanoic acid. Synthesis, resolution, and effects on carnitine acyltransferases.EBI
University of Alabama At Birmingham
Synthesis, biological assay in vitro and molecular docking studies of new Schiff base derivatives as potential urease inhibitors.EBI
Comsats Institute of Information Technology
Enzyme inhibitory activities an insight into the structure-Activity relationship of biscoumarin derivatives.EBI
Quaid-I-Azam University
Design and synthesis of a potent and selective triazolone-based peroxisome proliferator-activated receptor alpha agonist.EBI
Eli Lilly
Synthesis of biphenyl oxazole derivatives via Suzuki coupling and biological evaluations as nucleotide pyrophosphatase/phosphodiesterase-1 and -3 inhibitors.EBI
Quaid-I-Azam University
Developing new hybrid scaffold for urease inhibition based on carbazole-chalcone conjugates: Synthesis, assessment of therapeutic potential and computational docking analysis.EBI
Quaid-I-Azam University
Hydroxyl substituted benzoic acid/cinnamic acid derivatives: Tyrosinase inhibitory kinetics, anti-melanogenic activity and molecular docking studies.EBI
The University of Queensland (Uq)
Exploration of carboxy pyrazole derivatives: Synthesis, alkaline phosphatase, nucleotide pyrophosphatase/phosphodiesterase and nucleoside triphosphate diphosphohydrolase inhibition studies with potential anticancer profile.EBI
Quaid-I-Azam University
Design, synthesis, kinetic mechanism and molecular docking studies of novel 1-pentanoyl-3-arylthioureas as inhibitors of mushroom tyrosinase and free radical scavengers.EBI
Quaid-I-Azam University
Synthesis of sulfadiazinyl acyl/aryl thiourea derivatives as calf intestinal alkaline phosphatase inhibitors, pharmacokinetic properties, lead optimization, Lineweaver-Burk plot evaluation and binding analysis.EBI
Quaid-I-Azam University
CYCLIC AMINE DERIVATIVES HAVING SEROTONIN RECEPTOR BINDING ACTIVITYBDB
Shionogi
Factor IXa inhibitorsBDB
Merck Sharp & Dohme
Meta-substituted phenyl sulfonyl amides of secondary amino acid amides, the production thereof, and use thereof as matriptase inhibitorsBDB
The Medicines Company (Leipzig)
6,7-unsaturated-7-carbamoyl substituted morphinan derivativeBDB
Shionogi
Synthesis and in vitro opioid activity profiles of DALDA analogues.BDB
Clinical Research Institute of Montreal
Characterization of human A(2B) adenosine receptors: radioligand binding, western blotting, and coupling to G(q) in human embryonic kidney 293 cells and HMC-1 mast cells.BDB
University of Virginia