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10 articles for DR Jakas


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
15
Discovery of an imidazopyridine-containing 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonist with efficacy in a restenosis model.EBI
Smithkline Beecham Pharmaceuticals
17
 
Structure-activity relationships in 3-oxo-1,4-benzodiazepine-2-acetic acid GPIIb/IIIa antagonists. The 2-benzazepine seriesEBI
TBA
5
Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model.EBI
Smithkline Beecham Pharmaceuticals
21
Conformational preferences in a benzodiazepine series of potent nonpeptide fibrinogen receptor antagonists.EBI
Smithkline Beecham Pharmaceuticals
40
Benzimidazole derivatives as arginine mimetics in 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonists.EBI
Smithkline Beecham Pharmaceuticals
10
Potent, selective, orally active 3-oxo-1,4-benzodiazepine GPIIb/IIIa integrin antagonists.EBI
Smithkline Beecham Pharmaceuticals
6
(E)-3-[[[[6-(2-carboxyethenyl)-5-[[8-(4- methoxyphenyl)octyl]oxy]-2-pyridinyl]-methyl]thio]methyl]benzoic acid: a novel high-affinity leukotriene B4 receptor antagonist.EBI
Smithkline Beecham Pharmaceuticals
32
Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships.EBI
Smithkline Beecham Pharmaceuticals
19
(E)-3-[[[[6-(2-carboxyethenyl)-5-[[8-(4- methoxyphenyl)octyl]oxy]-2-pyridinyl]-methyl]thio]methyl]benzoic acid and related compounds: high affinity leukotriene B4 receptor antagonists.EBI
Smithkline Beecham Pharmaceuticals
35
Nonpeptide cyclic cyanoguanidines as HIV-1 protease inhibitors: synthesis, structure-activity relationships, and X-ray crystal structure studies.BDB
Dupont Pharmaceuticals