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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 745K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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13 articles for Y Koh


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Reduction of peptide character of HIV protease inhibitors that exhibit nanomolar potency against multidrug resistant HIV-1 strains.EBI
Kyoto University
Discovery of Leucyladenylate Sulfamates as Novel Leucyl-tRNA Synthetase (LRS)-Targeted Mammalian Target of Rapamycin Complex 1 (mTORC1) Inhibitors.EBI
Seoul National University
Design and synthesis of potent HIV-1 protease inhibitors incorporating hexahydrofuropyranol-derived high affinity P(2) ligands: structure-activity studies and biological evaluation.EBI
Purdue University
Synthesis and biological evaluation of novel allophenylnorstatine-based HIV-1 protease inhibitors incorporating high affinity P2-ligands.EBI
Purdue University
Potent inhibition of HIV-1 replication by novel non-peptidyl small molecule inhibitors of protease dimerization.EBI
Kumamoto University Graduate School of Medical and Pharmaceutical Sciences
Discovery of simplified leucyladenylate sulfamates as novel leucyl-tRNA synthetase (LRS)-targeted mammalian target of rapamycin complex 1 (mTORC1) inhibitors.EBI
Seoul National University
Compounds and compositions as RAF kinase inhibitorsBDB
Novartis
Keto-imidazopyridine derivatives as RORc modulatorsBDB
Genentech
2-(morpholin-4-yl)-1,7-naphthyridinesBDB
Bayer Pharma Aktiengesellschaft
Differences in the central nervous system distribution and pharmacology of the mouse 5-hydroxytryptamine-6 receptor compared with rat and human receptors investigated by radioligand binding, site-directed mutagenesis, and molecular modeling.BDB
Glaxosmithkline
Discovery of potent antagonists of the antiapoptotic protein XIAP for the treatment of cancer.BDB
Abbott Laboratories
Structure-based design of caspase-1 inhibitor containing a diphenyl ether sulfonamide.BDB
Pfizer
New anilinophthalazines as potent and orally well absorbed inhibitors of the VEGF receptor tyrosine kinases useful as antagonists of tumor-driven angiogenesis.BDB
Novartis Pharmaceuticals