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20 articles for FM Sirotnak


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
6
Synthesis and biological evaluation of 8-deazahomofolic acid and its tetrahydro derivative.EBI
Sri International
10
Syntheses and antifolate activity of 5-methyl-5-deaza analogues of aminopterin, methotrexate, folic acid, and N10-methylfolic acid.EBI
TBA
5
10-Propargylaminopterin and alkyl homologues of methotrexate as inhibitors of folate metabolism.EBI
TBA
6
Synthesis and antitumor activity of 10-alkyl-10-deazaminopterins. A convenient synthesis of 10-deazaminopterin.EBI
TBA
7
Synthesis and antitumor activity of 10-propargyl-10-deazaaminopterin.EBI
Sri International
10
Studies on analogues of classical antifolates bearing the naphthoyl group in place of benzoyl in the side chain.EBI
Southern Research Institute
13
Syntheses of alpha- and gamma-substituted amides, peptides, and esters of methotrexate and their evaluation as inhibitors of folate metabolism.EBI
TBA
7
Folate analogues altered in the C9-N10 bridge region. 18. Synthesis and antitumor evaluation of 11-oxahomoaminopterin and related compounds.EBI
TBA
3
Folate analogues. 21. Synthesis and antifolate and antitumor activities of N10-(cyanomethyl)-5,8-dideazafolic acid.EBI
TBA
25
9-substituted acridine derivatives with long half-life and potent antitumor activity: synthesis and structure-activity relationships.EBI
Sloan-Kettering Institute For Cancer Research
10
Syntheses and evaluation as antifolates of MTX analogues derived from 2, omega-diaminoalkanoic acids.EBI
TBA
9
Synthesis and biological activity of resolved C-10 diastereomers of 10-methyl- and 10-ethyl-10-deazaminopterin.EBI
TBA
7
Chemical synthesis and biological activities of 5-deazaaminopterin analogues bearing substituent(s) at the 5- and/or 7-position(s).EBI
Cornell University
5
Synthesis and antifolate activity of 5-methyl-5,10-dideaza analogues of aminopterin and folic acid and an alternative synthesis of 5,10-dideazatetrahydrofolic acid, a potent inhibitor of glycinamide ribonucleotide formyltransferase.EBI
Southern Research Institute
3
Synthesis and antifolate properties of 5,10-methylenetetrahydro-8,10-dideazaminopterin.EBI
TBA
6
Synthesis and antifolate properties of 10-alkyl-5,10-dideaza analogues of methotrexate and tetrahydrofolic acid.EBI
Sri International
5
Synthesis and antifolate properties of 9-alkyl-10-deazaminopterins.EBI
Sri International
6
Synthesis and antifolate evaluation of the 10-propargyl derivatives of 5-deazafolic acid, 5-deazaaminopterin, and 5-methyl-5-deazaaminopterin.EBI
Southern Research Institute
4
Synthesis and antifolate properties of 5,10-ethano-5,10-dideazaaminopterin.EBI
Sri International
2
Synthesis and antifolate evaluation of 10-ethyl-5-methyl-5,10- dideazaaminopterin and an alternative synthesis of 10-ethyl-10- deazaaminopterin (edatrexate).EBI
Southern Research Institute