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20 articles for Z Yuan


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of Fluorine-Containing Benzoxazinyl-oxazolidinones for the Treatment of Multidrug Resistant Tuberculosis.EBI
Peking Union Medical College
Exploiting the P-1 pocket of BRCT domains toward a structure guided inhibitor design.EBI
TBA
Structure-activity relationship studies to probe the phosphoprotein binding site on the carboxy terminal domains of the breast cancer susceptibility gene 1.EBI
University of Nebraska Medical Center
 
Novel indolactam-based inhibitors of matrix metalloproteinasesEBI
TBA
Discovery of novel nucleoside derivatives as selective lysine acetyltransferase p300 inhibitors for cancer therapy.EBI
Changsha Medical University
Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A Inhibitors.EBI
Nanjing University of Chinese Medicine
Discovery of C-3 isoxazole substituted thiochromone S,S-dioxide derivatives as potent and selective inhibitors for monoamine oxidase B (MAO-B).EBI
University of South China
Optimization, and biological evaluation of 3-O-β-chacotriosyl betulinic acid amide derivatives as novel small-molecule Omicron.EBI
South China Agricultural University
Inhibition of GABA shunt enzymes' activity by 4-hydroxybenzaldehyde derivatives.EBI
Huazhong University of Science and Technology
Quinazoline-based hydroxamic acid derivatives as dual histone methylation and deacetylation inhibitors for potential anticancer agents.EBI
Tsinghua University
Discovery of a novel small-molecule inhibitor of Fam20C that induces apoptosis and inhibits migration in triple negative breast cancer.EBI
Southwest Jiaotong University
Design, synthesis and evaluation of novel ErbB/HDAC multitargeted inhibitors with selectivity in EGFREBI
Tsinghua University
Discovery of triazolo [1,5-a] pyridine derivatives as novel JAK1/2 inhibitors.EBI
Shenyang Pharmaceutical University
Exploring structure-activity relationships around the phosphomannose isomerase inhibitor AF14049 via combinatorial synthesis.EBI
Affymax Research Institute
Discovery of a Novel Selective Dual Peroxisome Proliferator-Activated Receptor α/δ Agonist for the Treatment of Primary Biliary Cirrhosis.EBI
Wuxi Apptec (Shanghai) Co.
Design, synthesis and anticancer evaluation of acridine hydroxamic acid derivatives as dual Topo and HDAC inhibitors.EBI
Tsinghua University
Phthalimide conjugations for the degradation of oncogenic PI3K.EBI
Tsinghua University
Design, synthesis and biological evaluation of 4-amidobenzimidazole acridine derivatives as dual PARP and Topo inhibitors for cancer therapy.EBI
Tsinghua University
Olaparib hydroxamic acid derivatives as dual PARP and HDAC inhibitors for cancer therapy.EBI
Tsinghua University
Design, synthesis and anticancer potential of NSC-319745 hydroxamic acid derivatives as DNMT and HDAC inhibitors.EBI
Tsinghua University