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21 articles for L Naesens


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Virtual Screening and Biological Validation of Novel Influenza Virus PA Endonuclease Inhibitors.EBI
University of Sassari
Antimalarial activity of prodrugs of N-branched acyclic nucleoside phosphonate inhibitors of 6-oxopurine phosphoribosyltransferases.EBI
Academy of Sciences of The Czech Republic
New polycyclic dual inhibitors of the wild type and the V27A mutant M2 channel of the influenza A virus with unexpected binding mode.EBI
Universitat De Barcelona
Aza-acyclic nucleoside phosphonates containing a second phosphonate group as inhibitors of the human, Plasmodium falciparum and vivax 6-oxopurine phosphoribosyltransferases and their prodrugs as antimalarial agents.EBI
The University of Queensland
Azapropellanes with anti-influenza a virus activity.EBI
Universitat De Barcelona
Norbornane-based nucleoside and nucleotide analogues locked in North conformation.EBI
Academy of Sciences of The Czech Republic
Easily accessible polycyclic amines that inhibit the wild-type and amantadine-resistant mutants of the M2 channel of influenza A virus.EBI
Universitat De Barcelona
Acyclic nucleoside phosphonates containing a second phosphonate group are potent inhibitors of 6-oxopurine phosphoribosyltransferases and have antimalarial activity.EBI
The University of Queensland
Microwave assisted synthesis and anti-influenza virus activity of 1-adamantyl substituted N-(1-thia-4-azaspiro[4.5]decan-4-yl)carboxamide derivatives.EBI
Istanbul University
Exploring the size limit of templates for inhibitors of the M2 ion channel of influenza A virus.EBI
Universitat De Barcelona
Xanthine-Guanine-Hypoxanthine Phosphoribosyltransferase-A Putative Target for Drug Discovery against Gastrointestinal Tract Infections.EBI
The University of Queensland
N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interaction.EBI
Instituto De Qu£Mica M£Dica (C.S.I.C.)
Bicyclic α-Iminophosphonates as High Affinity Imidazoline IEBI
University of Barcelona
1,6-Bis[(benzyloxy)methyl]uracil derivatives-Novel antivirals with activity against HIV-1 and influenza H1N1 virus.EBI
Volgograd State Medical University
3-Azatetracyclo[5.2.1.1(5,8).0(1,5)]undecane derivatives: from wild-type inhibitors of the M2 ion channel of influenza A virus to derivatives with potent activity against the V27A mutant.EBI
Universitat De Barcelona
Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening.EBI
Polo Universitario Ss. Annunziata
Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR).EBI
University of Genoa
Synthesis and evaluation of symmetric acyclic nucleoside bisphosphonates as inhibitors of the Plasmodium falciparum, Plasmodium vivax and human 6-oxopurine phosphoribosyltransferases and the antimalarial activity of their prodrugs.EBI
The Institute of Organic Chemistry and Biochemistry of The Czech Academy of Sciences
Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus.EBI
University of Genoa
Slow but Steady Wins the Race: Dissimilarities among New Dual Inhibitors of the Wild-Type and the V27A Mutant M2 Channels of Influenza A Virus.EBI
Universitat De Barcelona
Synthesis and Evaluation of Asymmetric Acyclic Nucleoside Bisphosphonates as Inhibitors of Plasmodium falciparum and Human Hypoxanthine-Guanine-(Xanthine) Phosphoribosyltransferase.EBI
The Institute of Organic Chemistry and Biochemistry of The Czech Academy of Sciences