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22 articles for BT Berger


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2.EBI
Goethe University Frankfurt
NVP-BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family.EBI
Johann Wolfgang Goethe University
Discovery of Two Highly Selective Structurally Orthogonal Chemical Probes for Activin Receptor-like Kinases 1 and 2.EBI
Johann Wolfgang Goethe-University
Back-Pocket Optimization of 2-Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors.EBI
Goethe University
Synthesis of Pyrazole-Based Macrocycles Leads to a Highly Selective Inhibitor for MST3.EBI
Goethe University Frankfurt
Development of Selective Pyrido[2,3-d]pyrimidin-7(8H)-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors.EBI
Goethe University Frankfurt
MSC-1186, a Highly Selective Pan-SRPK Inhibitor Based on an Exceptionally Decorated Benzimidazole-Pyrimidine Core.EBI
Goethe University Frankfurt
Design and Synthesis of Pyrazole-Based Macrocyclic Kinase Inhibitors Targeting BMPR2.EBI
Johann Wolfgang Goethe-University
Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5-EBI
Goethe University Frankfurt
Design of a "Two-in-One" Mutant-Selective Epidermal Growth Factor Receptor Inhibitor That Spans the Orthosteric and Allosteric Sites.EBI
Eberhard Karls Universit£T T£Bingen
Structure-Based Design of Selective Salt-Inducible Kinase Inhibitors.EBI
Johann Wolfgang Goethe University
Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes.EBI
Johann Wolfgang Goethe-University
Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe.EBI
Johann Wolfgang Goethe University
Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold.EBI
University of Campinas (Unicamp)
Design and Development of a Chemical Probe for Pseudokinase CaEBI
Goethe University Frankfurt Am Main
Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core.EBI
Masaryk University
Selective targeting of the αC and DFG-out pocket in p38 MAPK.EBI
Johann Wolfgang Goethe University
Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor.EBI
Goethe University Frankfurt
Bioisosteric Replacement of Arylamide-Linked Spine Residues with EBI
Federal University of Rio De Janeiro (Ufrj)
SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK).EBI
Johann Wolfgang Goethe University
Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors.EBI
Johann Wolfgang Goethe-University
Development, Optimization, and Structure-Activity Relationships of Covalent-Reversible JAK3 Inhibitors Based on a Tricyclic Imidazo[5,4- d]pyrrolo[2,3- b]pyridine Scaffold.EBI
Eberhard Karls University T£Bingen