48 articles for G Rosse
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Macrocyclic Inhibitors of ERK2 Kinase.

Dart Neuroscience
Pyridyl Isonicotinamide Inhibitors of RAF Kinase.

Dart Neuroscience
Pyrazole Inhibitors of GluN2B NMDA Receptor Subunit.

Dart Neuroscience
Quinazoline Carboxamides as Selective Antagonists of Adenosine 2A Receptor.

Dart Neuroscience
Imidazopyridazine Inhibitors of PI3Kß.

Dart Neuroscience
Dihydropteridinone Inhibitors of BRD4.

Dart Neuroscience
Pyridinonaphthyridinone Inhibitors of Type 2 Methionine Aminopeptidase.

Dart Neuroscience
Novel Pyridyloxadiazole Agonists of Sphingosin-1-phosphate.

Dart Neuroscience
Novel Disubstituted Pyrimidines as Inhibitors of Bruton's Tyrosine Kinase.

Dart Neuroscience
Pyrrolopyridines-quinazolines Inhibitors of PKR-Like ER Kinase.

Dart Neuroscience
Novel azaindazole sulfonamides inhibitors of serum and glucocorticoid regulated kinase.

Dart Neuroscience
Quinalozinones as Inhibitors of Class I PI3K Kinases.

Dart Neuroscience
Pyrrolopyrimidine Analogues as MKNK Inhibitors.

Dart Neuroscience
Combination of novel imidazopyridazine mps-1 kinase inhibitors and bcl-2 family protein inhibitors.

Dart Neuroscience
Pyrazolsulfonamide agonists of oxytocin receptor.

Dart Neuroscience
Triazolo[4,5-d]pyrimidine Derivatives as Inhibitors of GCN2.

Dart Neuroscience
Novel cycloalkenepyrazoles as inhibitors of bub1 kinase.

Dart Neuroscience
Phenyl carboxamide analogues as spleen tyrosine kinase (syk) inhibitors.

Dart Neuroscience
Thiazolocarboxamide Analogues as NAMPT Inhibitors.

Dart Neuroscience
Quinoline Derivatives as 5-HT6 Receptor PET Ligands.

Dart Neuroscience
Trisubstituted imidazoles as positive modulators of metabotropic glutamate receptor subtype 5.

Dart Neuroscience
Tricyclic Pyrimidines As Inhibitors of DYRK1A/DYRK1B As Potential Treatment for Down's Syndrome or Alzheimer's Disease.

Dart Neuroscience
Novel thiazolobenzodiazepines as inhibitors of histamine h3 receptor.

Dart Neuroscience
Positive allosteric modulators of nicotinic acetylcholine receptor.

Dart Neuroscience
Irreversible inhibitors of cysteine proteases.

Dart Neuroscience
Modulators of the GPR119 Receptor for the Treatment of Metabolic Syndrome.

Dart Neuroscience
Metabolites of the pyrimidine amine preladenant as adenosine a2a receptor antagonists.

Dart Neuroscience
Phenyl-quinoline-xxo-butyric Acid Inhibitors of Histone Lysine Demethylase for the Treatment of Cancer.

Arrival Discovery
Novel Pyrazolopyridine Inhibitors of Monoacylglycerol Lipase for the Treatment of Neurodegenerative Diseases and Neuroinflammation.

Arrival Discovery
Spiro-naphthyridine Antagonists of the Melanocortin Receptor 4 for the Treatment of Cachexia Associated with Chronic Illness.

Arrival Discovery
Amino-cyclohexane Carboxylic Acid Inhibitors of Arginase.

Arrival Discovery
Pyrazolidine Carboxamide Analogs as Selective Agonists of the Cannabinoid 2 Receptor.

Arrival Discovery
A Series of Pyrazole Analogs Binding to KRASG12C as Potential Cancer Treatment.

Arrival Discovery
Aminotriazole and Aminotetrazole Inhibitors of LSD1 as Epigenetic Modulators.

Dart Neuroscience
Treatment of Pain with Spirocylic Cyclohexane Derivatives Having Dual Specificity for ORL-1 and μ-Opioid Receptors.

Dart Neuroscience
Novel Pyrazolyl-dihydroisoquinolines as Positive Allosteric Modulator of the Dopamine D1 Receptor.

Arrival Discovery
Novel Methyl-aza-quinazolines as Inhibitors of the RAS-SOS Interaction.

Arrival Discovery
Novel Bis-heteroaryl Derivatives To Modulate Protein Aggregation for the Treatment of Neurodegenerative Diseases.

Drexel University
Imidazoquinolines as Novel Inhibitors of LRRK2 Kinase Activity.

Drexel University
Diazaspirononane Inhibitors of O-GlcNAc Hydrolase for the Treatment of Central Nervous System Diseases.

Drexel University
Diphenylpropane Derivatives as Agonist of PPAR Nuclear Receptors.

Dart Neuroscience
Anabaseine analogues as modulators of nicotinic acetylcholine receptor.

Dart Neuroscience
Imidazopyrazine Derivatives As Inhibitors of mTOR.

Dart Neuroscience
Negative allosteric modulators of metabotropic glutamate receptor subtype.

Dart Neuroscience
Dihydrooxazines As Inhibitors of BACE-1 or BACE-2.

Dart Neuroscience
Novel and selective inhibitors of histone deacetylase: patent highlight.

Dart Neuroscience
Benzenesulfonyl and Benzenesulfonamide as Modulators of the 5-HT6 Receptor: Patent Highlight.

Dart Neuroscience
Indolinone Inhibitors of ENT1 for the Treatment of Schizophrenia.

Dart Neuroscience