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48 articles for G Rosse


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Macrocyclic Inhibitors of ERK2 Kinase.EBI
Dart Neuroscience
Pyridyl Isonicotinamide Inhibitors of RAF Kinase.EBI
Dart Neuroscience
Pyrazole Inhibitors of GluN2B NMDA Receptor Subunit.EBI
Dart Neuroscience
Quinazoline Carboxamides as Selective Antagonists of Adenosine 2A Receptor.EBI
Dart Neuroscience
Imidazopyridazine Inhibitors of PI3Kß.EBI
Dart Neuroscience
Dihydropteridinone Inhibitors of BRD4.EBI
Dart Neuroscience
Pyridinonaphthyridinone Inhibitors of Type 2 Methionine Aminopeptidase.EBI
Dart Neuroscience
Novel Pyridyloxadiazole Agonists of Sphingosin-1-phosphate.EBI
Dart Neuroscience
Novel Disubstituted Pyrimidines as Inhibitors of Bruton's Tyrosine Kinase.EBI
Dart Neuroscience
Pyrrolopyridines-quinazolines Inhibitors of PKR-Like ER Kinase.EBI
Dart Neuroscience
Novel azaindazole sulfonamides inhibitors of serum and glucocorticoid regulated kinase.EBI
Dart Neuroscience
Quinalozinones as Inhibitors of Class I PI3K Kinases.EBI
Dart Neuroscience
Pyrrolopyrimidine Analogues as MKNK Inhibitors.EBI
Dart Neuroscience
Combination of novel imidazopyridazine mps-1 kinase inhibitors and bcl-2 family protein inhibitors.EBI
Dart Neuroscience
Pyrazolsulfonamide agonists of oxytocin receptor.EBI
Dart Neuroscience
Triazolo[4,5-d]pyrimidine Derivatives as Inhibitors of GCN2.EBI
Dart Neuroscience
Novel cycloalkenepyrazoles as inhibitors of bub1 kinase.EBI
Dart Neuroscience
Phenyl carboxamide analogues as spleen tyrosine kinase (syk) inhibitors.EBI
Dart Neuroscience
Thiazolocarboxamide Analogues as NAMPT Inhibitors.EBI
Dart Neuroscience
Quinoline Derivatives as 5-HT6 Receptor PET Ligands.EBI
Dart Neuroscience
Trisubstituted imidazoles as positive modulators of metabotropic glutamate receptor subtype 5.EBI
Dart Neuroscience
Tricyclic Pyrimidines As Inhibitors of DYRK1A/DYRK1B As Potential Treatment for Down's Syndrome or Alzheimer's Disease.EBI
Dart Neuroscience
Novel thiazolobenzodiazepines as inhibitors of histamine h3 receptor.EBI
Dart Neuroscience
Positive allosteric modulators of nicotinic acetylcholine receptor.EBI
Dart Neuroscience
Irreversible inhibitors of cysteine proteases.EBI
Dart Neuroscience
Modulators of the GPR119 Receptor for the Treatment of Metabolic Syndrome.EBI
Dart Neuroscience
Metabolites of the pyrimidine amine preladenant as adenosine a2a receptor antagonists.EBI
Dart Neuroscience
Phenyl-quinoline-xxo-butyric Acid Inhibitors of Histone Lysine Demethylase for the Treatment of Cancer.EBI
Arrival Discovery
Novel Pyrazolopyridine Inhibitors of Monoacylglycerol Lipase for the Treatment of Neurodegenerative Diseases and Neuroinflammation.EBI
Arrival Discovery
Spiro-naphthyridine Antagonists of the Melanocortin Receptor 4 for the Treatment of Cachexia Associated with Chronic Illness.EBI
Arrival Discovery
Amino-cyclohexane Carboxylic Acid Inhibitors of Arginase.EBI
Arrival Discovery
Pyrazolidine Carboxamide Analogs as Selective Agonists of the Cannabinoid 2 Receptor.EBI
Arrival Discovery
A Series of Pyrazole Analogs Binding to KRASG12C as Potential Cancer Treatment.EBI
Arrival Discovery
Aminotriazole and Aminotetrazole Inhibitors of LSD1 as Epigenetic Modulators.EBI
Dart Neuroscience
Treatment of Pain with Spirocylic Cyclohexane Derivatives Having Dual Specificity for ORL-1 and μ-Opioid Receptors.EBI
Dart Neuroscience
Novel Pyrazolyl-dihydroisoquinolines as Positive Allosteric Modulator of the Dopamine D1 Receptor.EBI
Arrival Discovery
Novel Methyl-aza-quinazolines as Inhibitors of the RAS-SOS Interaction.EBI
Arrival Discovery
Novel Bis-heteroaryl Derivatives To Modulate Protein Aggregation for the Treatment of Neurodegenerative Diseases.EBI
Drexel University
Imidazoquinolines as Novel Inhibitors of LRRK2 Kinase Activity.EBI
Drexel University
Diazaspirononane Inhibitors of O-GlcNAc Hydrolase for the Treatment of Central Nervous System Diseases.EBI
Drexel University
Diphenylpropane Derivatives as Agonist of PPAR Nuclear Receptors.EBI
Dart Neuroscience
Anabaseine analogues as modulators of nicotinic acetylcholine receptor.EBI
Dart Neuroscience
Imidazopyrazine Derivatives As Inhibitors of mTOR.EBI
Dart Neuroscience
Negative allosteric modulators of metabotropic glutamate receptor subtype.EBI
Dart Neuroscience
Dihydrooxazines As Inhibitors of BACE-1 or BACE-2.EBI
Dart Neuroscience
Novel and selective inhibitors of histone deacetylase: patent highlight.EBI
Dart Neuroscience
Benzenesulfonyl and Benzenesulfonamide as Modulators of the 5-HT6 Receptor: Patent Highlight.EBI
Dart Neuroscience
Indolinone Inhibitors of ENT1 for the Treatment of Schizophrenia.EBI
Dart Neuroscience