The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 756K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

To help with training and testing AI and other models, BindingDB downloads and search results now provide the publication date and BindingDB curation date of each measurement.

19 articles for I Bruno


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis, in vitro evaluation, and molecular modeling investigation of benzenesulfonimide peroxisome proliferator-activated receptorsa antagonists.EBI
Universit£&Quot;G. D'Annunzio&Quot
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors.EBI
University of Salerno
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1).EBI
University of Salerno
Identification of new¿-hydroxybutenolides that preferentially inhibit the activity of mPGES-1.EBI
University of Salerno
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors.EBI
University of Salerno
Makaluvamine P, a new cytotoxic pyrroloiminoquinone from Zyzzya cf. fuliginosa.EBI
University of Salerno
Structure-based discovery of inhibitors of microsomal prostaglandin E2 synthase-1, 5-lipoxygenase and 5-lipoxygenase-activating protein: promising hits for the development of new anti-inflammatory agents.EBI
University of Salerno
Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222.EBI
University of Salerno
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders.EBI
University of Salerno
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin EEBI
University of Salerno
Discovery of noscapine derivatives as potential β-tubulin inhibitors.EBI
Shahid Beheshti University
Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking Studies.EBI
"G. D'Annunzio" University of Chieti-Pescara
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGEEBI
University of Salerno
Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition.EBI
Institute of Biomolecular Chemistry (Icb)
Novel Phenyldiazenyl Fibrate Analogues as PPAR α/γ/δ Pan-Agonists for the Amelioration of Metabolic Syndrome.EBI
University of Chieti "G. D.Annunzio
Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors.EBI
University of Salerno
Polycyclic guanidine alkaloids from the marine sponge Crambe crambe and Ca++ channel blocker activity of crambescidin 816.EBI
University of Brussels
Discovery of new potent molecular entities able to inhibit mPGES-1.EBI
University of Salerno
Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors.EBI
University of Salerno