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23 articles for MP Giovannoni


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists.EBI
Universita Degli Studi Di Firenze
Optimization of N-benzoylindazole derivatives as inhibitors of human neutrophil elastase.EBI
Universita Degli Studi Di Firenze
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists.EBI
Universita Degli Studi Di Firenze
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase.EBI
Universita Degli Studi Di Firenze
Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A(1) adenosine receptor ligands.EBI
Dipartimento Di Scienze Farmaceutiche
Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain.EBI
Dipartimento Di Scienze Farmaceutiche
6-methyl-2,4-disubstituted pyridazin-3(2H)-ones: a novel class of small-molecule agonists for formyl peptide receptors.EBI
Universita Degli Studi Di Firenze
Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity.EBI
University of Florence
4-Amino-5-vinyl-3(2H)-pyridazinones and analogues as potent antinociceptive agents: Synthesis, SARs, and preliminary studies on the mechanism of action.EBI
Dipartimento Di Scienze Farmaceutiche
Arylpiperazinylalkylpyridazinones and analogues as potent and orally active antinociceptive agents: synthesis and studies on mechanism of action.EBI
Dipartimento Di Scienze Farmaceutiche
Novel pyrazolopyrimidopyridazinones with potent and selective phosphodiesterase 5 (PDE5) inhibitory activity as potential agents for treatment of erectile dysfunction.EBI
Università
New pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective PDE5 inhibitors.EBI
RhôNe-Poulenc Rorer
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors.EBI
University of Florence
Design and synthesis of the first indole-based blockers of Panx-1 channel.EBI
University of Florence
Exploration of nitrogen heterocycle scaffolds for the development of potent human neutrophil elastase inhibitors.EBI
University of Florence
5,6-Diphenylpyridazine derivatives as acyl-CoA:cholesterol acyltransferase inhibitors.EBI
Università
Phenylpiperazinylalkylamino substituted pyridazinones as potent alpha(1) adrenoceptor antagonists.EBI
Istituto Chimico Farmaceutico E Tossicologico
Isoxazolo-[3,4-d]-pyridazin-7-(6H)-one as a potential substrate for new aldose reductase inhibitors.EBI
Dipartimento Di Scienze Farmaceutiche
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.EBI
Universita Degli Studi Di Firenze
Novel heterocyclic-fused pyridazinones as potent and selective phosphodiesterase IV inhibitors.EBI
Dipartimento Di Scienze Farmaceutiche, Firenze, Italy.
Presynaptic cholinergic modulators as potent cognition enhancers and analgesic drugs. 2. 2-Phenoxy-, 2-(phenylthio)-, and 2-(phenylamino)alkanoic acid esters.EBI
University of Florence
Presynaptic cholinergic modulators as potent cognition enhancers and analgesic drugs. 1. Tropic and 2-phenylpropionic acid esters.EBI
University of Florence
1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitors.EBI
University of Florence