18 articles for CA Maggi
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Lead optimization of P5U and urantide: discovery of novel potent ligands at the urotensin-II receptor.
University of Naples&Quot;Federico Ii&Quot
Design and synthesis of novel sulfonamide-containing bradykinin hB(2) receptor antagonists. Synthesis and structure-relationships ofa,a-tetrahydropyranylglycine.
Menarini Ricerche
hNK2 receptor antagonists. The use of intramolecular hydrogen bonding to increase solubility and membrane permeability.
Menarini Ricerche
Structure-activity relationships of 6-methyl-benzo[b]thiophene-2-carboxylic acid (1-[(S)-1-benzyl-4-[4-(tetrahydropyran-4-ylmethyl)piperazin-1-yl]butylcarbamoyl]cyclopentyl)amide, potent antagonist of the neurokinin-2 receptor.
Menarini Ricerche
New insight into the binding mode of peptide ligands at Urotensin-II receptor: structure-activity relationships study on P5U and urantide.
University of Naples Federico Ii
A new class of pseudopeptide antagonists of the kinin B1 receptor containing alkyl spacers.
Institute of Mutagenesis and Differentiation
Insertion of 2-carboxysuccinate and tricarballylic acid fragments into cyclic-pseudopeptides: new antagonists for the human tachykinin NK-2 receptor.
Menarini Ricerche S.P.A. Laboratori Di Firenze
Synthesis and biological activity of new bradykinin pseudopeptide B1 receptor agonists containing alkylic spacers
TBA
Benzofused hydroxamic acids: useful fragments for the preparation of histone deacetylase inhibitors. Part 1: hit identification.
Menarini Ricerche
Set-up of a new series of HDAC inhibitors: the 5,11-dihydrodibenzo[b,e]azepin-6-ones as privileged structures.
Menarini Ricerche Pomezia
4-N-Hydroxy-4-[1-(sulfonyl)piperidin-4-yl]-butyramides as HDAC inhibitors.
Menarini Ricerche Pomezia
Alkyl piperidine and piperazine hydroxamic acids as HDAC inhibitors.
Menarini Ricerche Pomezia
Antiproliferative and differentiating activities of a novel series of histone deacetylase inhibitors.
Menarini Ricerche
Discovery of a new series of potent and selective linear tachykinin NK2 receptor antagonists.
Menarini Ricerche
Insertion of an aspartic acid moiety into cyclic pseudopeptides: synthesis and biological characterization of potent antagonists for the human Tachykinin NK-2 receptor.
Menarini Ricerche
A new, potent urotensin II receptor peptide agonist containing a Pen residue at the disulfide bridge.
University of Naples Federico Ii
Monocyclic human tachykinin NK-2 receptor antagonists as evolution of a potent bicyclic antagonist: QSAR and site-directed mutagenesis studies.
Menarini Ricerche