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18 articles for R Gust


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Importance of 5/6-aryl substitution on the pharmacological profile of 4'-((2-propyl-1H-benzo[d]imidazol-1-yl)methyl)-[1,1'-biphenyl]-2-carboxylic acid derived PPAR¿ agonists.EBI
University of Innsbruck
Evaluation of selected 3D virtual screening tools for the prospective identification of peroxisome proliferator-activated receptor (PPAR)¿ partial agonists.EBI
University of Innsbruck
New telmisartan-derived PPAR¿ agonists: Impact of the 3D-binding mode on the pharmacological profile.EBI
Universit£T Innsbruck
Effects of C2-alkylation, N-alkylation, and N,N'-dialkylation on the stability and estrogen receptor interaction of (4R,5S)/(4S,5R)-4,5-bis(4-hydroxyphenyl)-2-imidazolines.EBI
Free University of Berlin
(4R,5S)/(4S,5R)-4,5-Bis(4-hydroxyphenyl)-2-imidazolines: ligands for the estrogen receptor with a novel binding mode.EBI
Free University of Berlin
Influence of chlorine or fluorine substitution on the estrogenic properties of 1-alkyl-2,3,5-tris(4-hydroxyphenyl)-1H-pyrroles.EBI
Freie Universit£T Berlin
2-phenyl-1-[4-(2-piperidine-1-yl-ethoxy)benzyl]-1H-benzimidazoles as ligands for the estrogen receptor: synthesis and pharmacological evaluation.EBI
Freie Universit£T Berlin
Target-based approach to inhibitors of histone arginine methyltransferases.EBI
Albert-Ludwigs-University of Freiburg
Characterization of new PPARgamma agonists: benzimidazole derivatives-importance of positions 5 and 6, and computational studies on the binding mode.EBI
Freie UniversitäT Berlin
Cobalt-alkyne complexes with imidazoline ligands as estrogenic carriers: synthesis and pharmacological investigations.EBI
Freie Universitat Berlin
Synthesis and pharmacological evaluation of 1H-imidazoles as ligands for the estrogen receptor and cytotoxic inhibitors of the cyclooxygenase.EBI
Free University of Berlin
Investigations on the effects of basic side chains on the hormonal profile of (4R,5S)/(4S,5R)-4,5-bis(4-hydroxyphenyl)-2-imidazolines.EBI
Free University of Berlin
Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site.EBI
University of Innsbruck
Identification and development of non-cytotoxic cell death modulators: Impact of sartans and derivatives on PPARγ activation and on growth of imatinib-resistant chronic myelogenous leukemia cells.EBI
University of Innsbruck
Investigations on estrogen receptor binding. The estrogenic, antiestrogenic, and cytotoxic properties of C2-alkyl-substituted 1,1-bis(4-hydroxyphenyl)-2-phenylethenes.EBI
Free University of Berlin
Development of bivalent triarylalkene- and cyclofenil-derived dual estrogen receptor antagonists and downregulators.EBI
University of Innsbruck
Overcoming imatinib resistance in chronic myelogenous leukemia cells using non-cytotoxic cell death modulators.EBI
University of Innsbruck
Antiestrogenically active 1,1,2-tris(4-hydroxyphenyl)alkenes without basic side chain: synthesis and biological activity.EBI
Free University of Berlin