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13 articles for G Colombo


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
57
Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile.EBI
Sapienza University of Rome
20
1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: an effective scaffold for the design of either CB1 or CB2 receptor ligands.EBI
Sapienza University of Rome
27
Synthesis and biological evaluation of new N-alkyl 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides as cannabinoid receptor ligands.EBI
Sapienza University of Rome
8
An efficient steroid pharmacophore-based strategy to identify new aromatase inhibitors.EBI
Universidade De Coimbra
88
Fast three dimensional pharmacophore virtual screening of new potent non-steroid aromatase inhibitors.EBI
Universidade De Coimbra
21
Design, Synthesis, and Physicochemical and Pharmacological Profiling of 7-Hydroxy-5-oxopyrazolo[4,3-EBI
University of Siena
7
Progress in the Field of Aldehyde Dehydrogenase Inhibitors: Novel Imidazo[1,2-EBI
University of Pisa
4
Dual Binding to Orthosteric and Allosteric Sites Enhances the Anticancer Activity of a TRAP1-Targeting Drug.EBI
Ulsan National Institutes of Science and Technology (Unist)
7
Rational design of allosteric modulators of the aromatase enzyme: An unprecedented therapeutic strategy to fight breast cancer.EBI
Cnr-Iom-Democritos C/O International School For Advanced Studies (Sissa)
18
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group.EBI
University of Pavia
13
Discovery of Highly Potent Benzimidazole Derivatives as Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors: From Structure-Based Virtual Screening to EBI
University of Eastern Piedmont
1
Allosteric Modulators of HSP90 and HSP70: Dynamics Meets Function through Structure-Based Drug Design.EBI
Istituto Di Chimica Del Riconoscimento Molecolare
11
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.EBI
The University of Kansas