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18 articles for CS Harris


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of novel TACE inhibitors compatible with topical application.EBI
Nestl�
Discovery of phenoxyindazoles and phenylthioindazoles as ROR¿ inverse agonists.EBI
Galderma R & D
Design of selective PI3Ka inhibitors starting from a promiscuous pan kinase scaffold.EBI
Astrazeneca
Structure-activity relationship of a series of non peptidic RGD integrin antagonists targetinga5ß1: part 1.EBI
Astrazeneca
Structure-activity relationship of a series of non peptidic RGD integrin antagonists targetinga5ß1: part 2.EBI
Astrazeneca
Synthesis and structure-activity relationships of thieno[2,3-b]pyrroles as antagonists of the GnRH receptor.EBI
Astrazeneca
Inhibitors of epidermal growth factor receptor tyrosine kinase: optimisation of potency and in vivo pharmacokinetics.EBI
Astrazeneca
Novel 4-anilinoquinazolines with C-6 carbon-linked side chains: synthesis and structure-activity relationship of a series of potent, orally active, EGF receptor tyrosine kinase inhibitors.EBI
Astrazeneca
Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket.EBI
Astrazeneca
Impact of Minor Structural Modifications on Properties of a Series of mTOR Inhibitors.EBI
Nestl�
Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma.EBI
Nestle Skin Health R&D
Sulfoximines as potent RORγ inverse agonists.EBI
Nestle Skin Health
New Caspase-1 inhibitor by scaffold hopping into bio-inspired 3D-fragment space.EBI
Edelris
Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis.EBI
Nestle Skin Health
Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne.EBI
Nestl�
Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors.EBI
Astrazeneca
The recent outbreaks of human coronaviruses: A medicinal chemistry perspective.BDB
University of Bonn
Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptor.BDB
University of Kansas