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14 articles for RA Engh


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of Aurora-A kinase.EBI
Evotec (Uk)
Crystal structures of catalytic subunit of cAMP-dependent protein kinase in complex with isoquinolinesulfonyl protein kinase inhibitors H7, H8, and H89. Structural implications for selectivity.EBI
Institute For Biochemistry
Tetrahydro-isoquinoline-based factor Xa inhibitors.EBI
Boehringer Mannheim
 
DERIVATIVES OF 4-AMINO-PYRIDINE AS SELECTIVE THROMBIN INHIBITORSEBI
TBA
In silico and NMR identification of inhibitors of the IGF-I and IGF-binding protein-5 interaction.EBI
Institute For Biochemistry
Probing the ATP-Binding Pocket of Protein Kinase DYRK1A with Benzothiazole Fragment Molecules.EBI
Uit The Arctic University of Norway
Novel acylguanidine containing thrombin inhibitors with reduced basicity at the P1 moiety.EBI
Nv Organon Scientific Development Group
Diarylsulfonamides as selective, non-peptidic thrombin inhibitors.EBI
Pharmazeutisch-Chemisches Institut Der UniversitäT
Bis-substituted malonic acid hydroxamate derivatives as inhibitors of human neutrophil collagenase (MMP8).EBI
Boehringer Mannheim
Novel Scaffolds for Dual Specificity Tyrosine-Phosphorylation-Regulated Kinase (DYRK1A) Inhibitors.EBI
Uit The Arctic University of Norway
γ-aminobutyric acid (GABA) analogues for the treatment of pain and other disordersBDB
Novassay
COMPOSITION CONTAINING ARYLAMIDE DERIVATIVEBDB
Chugai Seiyaku Kabushiki Kaisha
Identification of substituted 3-[(4,5,6, 7-tetrahydro-1H-indol-2-yl)methylene]-1,3-dihydroindol-2-ones as growth factor receptor inhibitors for VEGF-R2 (Flk-1/KDR), FGF-R1, and PDGF-Rbeta tyrosine kinases.BDB
Sugen
Tyrosine Kinase Inhibitors. 10. Isomeric 4-[(3-Bromophenyl)amino]pyrido[d]- pyrimidines Are Potent ATP Binding Site Inhibitors of the Tyrosine Kinase Function of the Epidermal Growth Factor ReceptorBDB
University of Auckland