25 articles for HR Kim
The following articles (labelled with PubMed ID or TBD) are for your review
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Replacing the terminal piperidine in ceritinib with aliphatic amines confers activities against crizotinib-resistant mutants including G1202R.

Korea Research Institute of Chemical Technology
Novel 2,4-diaminopyrimidines bearing tetrahydronaphthalenyl moiety against anaplastic lymphoma kinase (ALK): Synthesis, in vitro, ex vivo, and in vivo efficacy studies.

Chungbuk National University
Synthesis and evaluation of novel 2,4-diaminopyrimidines bearing bicyclic aminobenzazepines for anaplastic lymphoma kinase (ALK) inhibitor.

Korea Research Institute of Chemical Technology
Discovery of substituted 6-pheny-3H-pyridazin-3-one derivatives as novel c-Met kinase inhibitors.

Sungkyunkwan University
Design and synthesis of novel 3-(benzo[d]oxazol-2-yl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine derivatives as selective G-protein-coupled receptor kinase-2 and -5 inhibitors.

Korea Research Institute of Chemical Technology
Synthesis and structure-activity relationship of aminopyridines with substituted benzoxazoles as c-Met kinase inhibitors.

Korea Research Institute of Chemical Technology
Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitors.

Korea Research Institute of Chemical Technology
Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors.

Korea Research Institute of Chemical Technology
Design and synthesis of triazolopyridazines substituted with methylisoquinolinone as selective c-Met kinase inhibitors.

Korea Research Institute of Chemical Technology
Design, synthesis, and evaluation of 2-aryl-7-(3',4'-dialkoxyphenyl)-pyrazolo[1,5-a]pyrimidines as novel PDE-4 inhibitors.

Korea Research Institute of Chemical Technology
Structure-Activity Relationships of Truncated 1'-Homologated Carbaadenosine Derivatives as New PPARγ/δ Ligands: A Study on Sugar Puckering Affecting Binding to PPARs.

Seoul National University
Discovery of 2-aminoquinolone acid derivatives as potent inhibitors of SARS-CoV-2.

Seoul National University
Covalent Small Molecule Immunomodulators Targeting the Protease Active Site.

National Cancer Institute
Discovery of novel tetrahydroisoquinoline-containing pyrimidines as ALK inhibitors.

Korea Research Institute of Chemical Technology
Identification of 6'-β-fluoro-homoaristeromycin as a potent inhibitor of chikungunya virus replication.

Seoul National University
Design, Synthesis, and Anti-RNA Virus Activity of 6'-Fluorinated-Aristeromycin Analogues.

Seoul National University
Synthesis and biological evaluation of 3-acyl-2-phenylamino-1,4-dihydroquinolin-4(1H)-one derivatives as potential MERS-CoV inhibitors.

Korea Research Institute of Chemical Technology
Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase 1A (DYRK1A) Inhibitors as Potential Therapeutics.

Seoul National University
BACE1 inhibitory activity and molecular docking analysis of meroterpenoids from Sargassum serratifolium.

Pukyong National University
Novel 2,4-diaminopyrimidines bearing fused tricyclic ring moiety for anaplastic lymphoma kinase (ALK) inhibitor.

University of Science & Technology
Ethynyl derivatives

Hoffmann-La Roche
Bcl-2-selective apoptosis-inducing agents for the treatment of cancer and immune diseases

Abbvie
Bicyclic aryl and heteroaryl sodium channel inhibitors

Amgen
TRPV1 antagonists

TBA