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15 articles for J Dubois


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
New indolizine-chalcones as potent inhibitors of human farnesyltransferase: Design, synthesis and biological evaluation.EBI
Alexandru Ioan Cuza University
Studies on phenothiazines: New microtubule-interacting compounds with phenothiazine A-ring as potent antineoplastic agents.EBI
Alexandru Ioan Cuza University
Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors.EBI
Cnrs Upr2301
Novel indolizine derivatives with unprecedented inhibitory activity on human farnesyltransferase.EBI
Alexandru Ioan Cuza University
Chemical and biological explorations of the electrophilic reactivity of the bioactive marine natural product halenaquinone with biomimetic nucleophiles.EBI
University of Auckland
New bioactive halenaquinone derivatives from South Pacific marine sponges of the genus Xestospongia.EBI
National Museum of Natural History
Design and Synthesis of Tubulin and Histone Deacetylase Inhibitor Based on iso-Combretastatin A-4.EBI
Paris-Saclay University
Phenothiazine-based CaaX competitive inhibitors of human farnesyltransferase bearing a cysteine, methionine, serine or valine moiety as a new family of antitumoral compounds.EBI
Alexandru Ioan Cuza University
Synthesis and biological evaluation of a new series of N-ylides as protein farnesyltransferase inhibitors.EBI
'Al. I. Cuza' University of Iasi
Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors.EBI
Al. I. Cuza University of Iasi
Synthesis and biological evaluation of new phenothiazine derivatives bearing a pyrazole unit as protein farnesyltransferase inhibitors.EBI
'Al. I. Cuza' University of Iasi
New farnesyltransferase inhibitors in the phenothiazine series.EBI
Al. I. Cuza University of Iasi
Towards the synthesis of bisubstrate inhibitors of protein farnesyltransferase: Synthesis and biological evaluation of new farnesylpyrophosphate analogues.EBI
Centre De Recherche De Gif-Sur-Yvette
Macrocyclic compounds and their use as kinase inhibitorsBDB
Incyte
Chromenone derivativesBDB
Astrazeneca