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12 articles for P Grellier


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors.EBI
Cnrs Upr2301
Trends in research of antitrypanosomal agents among synthetic heterocycles.EBI
Danylo Halytsky Lviv National Medical University
Pharmacomodulation on the 3-acetylursolic acid skeleton: Design, synthesis, and biological evaluation of novel N-{3-[4-(3-aminopropyl)piperazinyl]propyl}-3-O-acetylursolamide derivatives as antimalarial agents.EBI
Universidade Federal Do Rio Grande Do Sul (Ufrgs)
Design, synthesis and in vitro antimalarial activity of an acylhydrazone library.EBI
University of Lille
Synthesis and in vitro and in vivo antimalarial activity of N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.EBI
University of Lille
Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives.EBI
University of Lille
Design, synthesis and antimalarial activity of novel, quinoline-based, zinc metallo-aminopeptidase inhibitors.EBI
University of Lille
Prolylisoxazoles: potent inhibitors of prolyloligopeptidase with antitrypanosomal activity.EBI
University of Antwerp
A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline.EBI
Umr 8525 Cnrs-Université
Automated parallel synthesis of a tetrahydroisoquinolin-based library: potential prolyl endopeptidase inhibitors.EBI
Université
Towards the synthesis of bisubstrate inhibitors of protein farnesyltransferase: Synthesis and biological evaluation of new farnesylpyrophosphate analogues.EBI
Centre De Recherche De Gif-Sur-Yvette
Macrocyclic compounds and their use as kinase inhibitorsBDB
Incyte