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26 articles for JL Gilmore


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of potent and selective nonsteroidal indazolyl amide glucocorticoid receptor agonists.EBI
Ironwood Pharmaceuticals
Synthesis and structure-activity relationships of novel indazolyl glucocorticoid receptor partial agonists.EBI
Bristol-Myers Squibb
A molecular modeling analysis of novel non-hydroxamate inhibitors of TACE.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Anilinodialkoxyquinazolines: screening epidermal growth factor receptor tyrosine kinase inhibitors for potential tumor imaging probes.EBI
Lawrence Berkeley National Laboratory
 
Synthesis and evaluation of 2-aryl-4H-3,1-benzoxazin-4-ones as C1r serine protease inhibitorsEBI
TBA
Synthesis and structure-activity relationship of a novel, non-hydroxamate series of TNF-alpha converting enzyme inhibitors.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Structure-activity relationship study of central pyridine-derived TYK2 JH2 inhibitors: Optimization of the PK profile through C4' and C6 variations.EBI
Bristol-Myers Squibb
Hydantoins, triazolones, and imidazolones as selective non-hydroxamate inhibitors of tumor necrosis factor-alpha converting enzyme (TACE).EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Discovery of novel hydantoins as selective non-hydroxamate inhibitors of tumor necrosis factor-alpha converting enzyme (TACE).EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Synthesis and structure-activity relationship of a novel, achiral series of TNF-alpha converting enzyme inhibitors.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Conversion of potent MMP inhibitors into selective TACE inhibitors.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Identification and Preclinical Pharmacology of ((1 R,3 S)-1-Amino-3-(( S)-6-(2-methoxyphenethyl)-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986166): A Differentiated Sphingosine-1-phosphate Receptor 1 (S1PEBI
Bristol-Myers Squibb Research and Development
Bicyclic Ligand-Biased Agonists of S1PEBI
Bristol Myers Squibb Research & Early Development
Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1PEBI
Bristol-Myers Squibb
Identification of Tricyclic Agonists of Sphingosine-1-phosphate Receptor 1 (S1PEBI
Bristol-Myers Squibb
Discovery and Structure-Activity Relationship (SAR) of a Series of Ethanolamine-Based Direct-Acting Agonists of Sphingosine-1-phosphate (S1P1).EBI
Bristol-Myers Squibb
Benzenesulfonamide derivatives of 2-substituted 4H-3,1-benzoxazin-4-ones and benzthiazin-4-ones as inhibitors of complement C1r protease.EBI
Warner-Lambert
2-amino-4H-3,1-benzoxazin-4-ones as inhibitors of C1r serine protease.EBI
Warner-Lambert
Method for preparing pyrrolidinyl urea derivativeBDB
Zhangzhou Pien Tze Huang Pharmaceutical
Inhibitors of RAF kinasesBDB
Kinnate Biopharma
TriazolopyrazineBDB
TBA
Substituted pyrrolo[1,2-b]pyridazines for treating disorders related to KIT and PDGFRBDB
Blueprint Medicines
Compounds as neuronal histamine receptor-3 antagonists and uses thereofBDB
Xw Laboratories
KCNQ2-5 channel activatorBDB
Ono Pharmaceutical
Substituted imidazopyrazinesBDB
Bayer Intellectual Property
Peripherally acting opioid compoundsBDB
Alkermes