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25 articles for Y Lv


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
23
Novel morpholin-3-one fused quinazoline derivatives as EGFR tyrosine kinase inhibitors.EBI
Beijing University of Technology
15
Design, synthesis, and biological activity of phenyl-pyrazole derivatives as BCR-ABL kinase inhibitors.EBI
Beijing University of Technology
27
Discovery of a New Series of Naphthamides as Potent VEGFR-2 Kinase Inhibitors.EBI
Chinese Academy of Sciences
5
Benzophenone C-glucosides and gallotannins from mango tree stem bark with broad-spectrum anti-viral activity.EBI
Chinese Academy of Sciences
2
Anti-inflammatory agents design via the fragment hybrid strategy in the discovery of compound c1 for treating ALI and UC.EBI
Wenzhou Medical University
21
Discovery of Novel Pyrrolo[2,3-b]pyridine-Based CSF-1R Inhibitors with Demonstrated Efficacy against Patient-Derived Colorectal Cancer Organoids.EBI
Nanjing University of Chinese Medicine
11
Recent advances in the development of dual ALK/ROS1 inhibitors for non-small cell lung cancer therapy.EBI
Weifang Medical University
9
Discovery of novel benzimidazole derivatives as selective and reversible monoamine oxidase B inhibitors for Parkinson's disease treatment.EBI
Zhejiang University
36
Discovery of a Novel CSF-1R Inhibitor with Highly Improved Pharmacokinetic Profiles and Superior Efficacy in Colorectal Cancer Immunotherapy.EBI
Nanjing University of Chinese Medicine
27
Discovery of C-3 isoxazole substituted thiochromone S,S-dioxide derivatives as potent and selective inhibitors for monoamine oxidase B (MAO-B).EBI
University of South China
2
A Potent SOS1 PROTAC Degrader with Synergistic Efficacy in Combination with KRASG12C Inhibitor.EBI
Ocean University of China
26
Design, synthesis and evaluation of C-5 substituted pyrrolopyridine derivatives as potent Janus Kinase 1 inhibitors with excellent selectivity.EBI
University of South China
3
Design, Construction, and Screening of Diversified Pyrimidine-Focused DNA-Encoded Libraries.EBI
Nanjing University of Chinese Medicine
31
Discovery of C-5 Pyrazole-Substituted Pyrrolopyridine Derivatives as Potent and Selective Inhibitors for Janus Kinase 1.EBI
University of South China
41
Rational Design, Synthesis, and Biological Evaluation of Novel S1PR2 Antagonists for Reversing 5-FU-Resistance in Colorectal Cancer.EBI
Ocean University of China
21
Design, synthesis and biological evaluation of sphingosine-1-phosphate receptor 2 antagonists as potent 5-FU-resistance reversal agents for the treatment of colorectal cancer.EBI
Laboratory For Marine Drugs and Bioproducts of Qingdao National Laboratory For Marine Science and Technology
13
Design, synthesis, and biological activity of 4-(imidazo[1,2-b]pyridazin-3-yl)-1H-pyrazol-1-yl-phenylbenzamide derivatives as BCR-ABL kinase inhibitors.EBI
Beijing University of Technology
27
Rational design, synthesis and biological evaluation of novel multitargeting anti-AD iron chelators with potent MAO-B inhibitory and antioxidant activity.EBI
Zhejiang University
3
Bioactivatable Pseudotripeptidization of Cyclic Dipeptides To Increase the Affinity toward Oligopeptide Transporter 1 for Enhanced Oral Absorption: An Application to Cyclo(l-Hyp-l-Ser) (JBP485).EBI
Dalian Medical University
31
Design, synthesis and biological evaluation of 1-hydroxy-2-phenyl-4-pyridyl-1H-imidazole derivatives as xanthine oxidase inhibitors.EBI
Shenyang Pharmaceutical University
20
Discovery of new thienopyrimidine derivatives as potent and orally efficacious phosphoinositide 3-kinase inhibitors.EBI
Peking Union Medical College
42
Discovery and Optimization of 2-Amino-4-methylquinazoline Derivatives as Highly Potent Phosphatidylinositol 3-Kinase Inhibitors for Cancer Treatment.EBI
Peking Union Medical College
1044
SARS-COV2 MAIN PROTEASE INHIBITORSBDB
Gilead Sciences
93
Naphthyridinone derivatives and their use in the treatment of arrhythmiaBDB
Novartis
4
Synthesis, inhibitory activity and molecular docking studies of two Cu(II) complexes against Helicobacter pylori urease.BDB
Wuhan Textile University