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25 articles for A Liang


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Designing allosteric regulators of thrombin. Monosulfated benzofuran dimers selectively interact with Arg173 of exosite 2 to induce inhibition.EBI
Virginia Commonwealth University
Solid-phase synthesis of naphthylamidines as factor VIIa/tissue factor inhibitors.EBI
Berlex Biosciences
Design, synthesis, and activity of a novel series of factor Xa inhibitors: optimization of arylamidine groups.EBI
Berlex Biosciences
Rational design of potent, small, synthetic allosteric inhibitors of thrombin.EBI
Virginia Commonwealth University
Discovery of novel and potent aryl diamines as leukotriene A4 hydrolase inhibitors.EBI
Berlex Biosciences
Synthesis of N-alkyl glycine amides as potent inhibitors of leukotriene A4 hydrolase.EBI
Berlex Biosciences
Synthesis and biological evaluation of piperazine-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1).EBI
Berlex Biosciences
Synthesis and biological evaluation of menthol-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1).EBI
Berlex Biosciences
Design and synthesis of aminophenol-based factor Xa inhibitors.EBI
Berlex Biosciences
Design, synthesis, and in vitro biological activity of benzimidazole based factor Xa inhibitors.EBI
Berlex Biosciences
Design, synthesis, and in vitro biological activity of indole-based factor Xa inhibitors.EBI
Berlex Biosciences
Synthesis, characterization, and structure-activity relationships of amidine-substituted (bis)benzylidene-cycloketone olefin isomers as potent and selective factor Xa inhibitors.EBI
Berlex Biosciences
Design, synthesis, and activity of 2,6-diphenoxypyridine-derived factor Xa inhibitors.EBI
Berlex Biosciences
Design, synthesis, and biological activity of novel purine and bicyclic pyrimidine factor Xa inhibitors.EBI
Berlex Biosciences
Solid-phase synthesis of N-substituted amidinophenoxy pyridines as factor XA inhibitors.EBI
Berlex Biosciences
Discovery of N-[2-[5-[Amino(imino)methyl]-2-hydroxyphenoxy]-3, 5-difluoro-6-[3-(4, 5-dihydro-1-methyl-1H-imidazol-2-yl)phenoxy]pyridin-4-yl]-N-methylgl y cine (ZK-807834): a potent, selective, and orally active inhibitor of the blood coagulation enzyme factor Xa.EBI
Berlex Biosciences
(Z,Z)-2,7-Bis(4-amidinobenzylidene)cycloheptan-1-one: identification of a highly active inhibitor of blood coagulation factor Xa.EBI
Berlex Biosciences
Identification of second-generation P2X3 antagonists for treatment of pain.EBI
Merck
Benzoxazolinone aryl sulfonamides as potent, selective NaEBI
Merck
1H-imidazo[4,5-h]quinazoline compound as protein kinase inhibitorBDB
Shengke Pharmaceuticals (Jiangsu)
PYRIDAZINYL AMINO DERIVATIVES AS ALK5 INHIBITORSBDB
Chiesi Farmaceutici
PHENYL TRIAZOLE MLL1-WDR5 PROTEIN-PROTEIN INTERACTION INHIBITORBDB
Huyabio International
Substituted pyrrolidines as factor XIa inhibitors for the treatment thromboembolic diseasesBDB
Ono Pharmaceutical
Substituted benzothiophenyl derivatives as GPR40 agonists for the treatment of type II diabetesBDB
Janssen Pharmaceutica
Benzimidazole derivatives as antihistamine agentsBDB
Faes Farma