43 articles for J Martinez
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Synthesis and biological activity of some partially modified retro-inverso analogues of cholecystokinin.
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Synthesis and biological activities of pseudopeptide analogues of the C-terminal heptapeptide of cholecystokinin. On the importance of the peptide bonds.
TBA
Imidazopyridine-fused [1,3]-diazepinones part 2: Structure-activity relationships and antiproliferative activity against melanoma cells.
University of Montpellier
New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center.
University of Montpellier
Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.
University of Montpellier
New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists.
University of Montpellier
Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.
University of Montpellier
Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT(7) and 5-HT(1A) receptor ligands.
Jagiellonian University Medical College
Fragment-based identification of a locus in the Sec7 domain of Arno for the design of protein-protein interaction inhibitors.
University of Montpellier
Further characterization of a putative serine protease contributing to the¿-secretase cleavage ofß-amyloid precursor protein.
University of Montpellier
Sulfonamides with the N-alkyl-N'-dialkylguanidine moiety as 5-HT7 receptor ligands.
Jagiellonian University Medical College
The influence of an ethylene spacer on the 5-HT(1A) and 5-HT(2A) receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones.
Jagiellonian University Medical College
Synthesis and characterization of bradykinin B(2) receptor agonists containing constrained dipeptide mimics.
University of Montpellier
Design and synthesis of potent bradykinin agonists containing a benzothiazepine moiety.
University of Montpellier
Structure-activity relationships of C-terminal tri- and tetrapeptide fragments that inhibit gastrin activity.
TBA
The design and synthesis of the high efficacy, non-peptide CCK1 receptor agonist PD170292.
Ccipe-Faculte De Pharmacie
Design, synthesis, and biological evaluation of 1,5-benzothiazepine-4-one derivatives targeting factor VIIa/tissue factor.
University of Montpellier
New trisubstituted 1,2,4-triazole derivatives as potent ghrelin receptor antagonists. 3. Synthesis and pharmacological in vitro and in vivo evaluations.
University of Montpellier
Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: on the significance of the orientation and substitution at position 3.
University of Montpellier
Synthesis and pharmacological in vitro and in vivo evaluations of novel triazole derivatives as ligands of the ghrelin receptor. 1.
University of Montpellier
Novel class of arylpiperazines containing N-acylated amino acids: their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation.
University of Montpellier
Arylpiperazines with N-acylated amino acids as 5-HT1A receptor ligands.
University of Montpellier
Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT
Jagiellonian University Medical College
A rational approach to the design and synthesis of a new bradykinin B(1) receptor antagonist.
University of Montpellier
Synthesis and biological evaluation of bradykinin B(1)/B(2) and selective B(1) receptor antagonists.
University of Montpellier
Synthesis and biological evaluation of bombesin constrained analogues.
University of Montpellier
Serotonin dimers: application of the bivalent ligand approach to the design of new potent and selective 5-HT(1B/1D) agonists.
Centre De Recherche Pierre Fabre
Cyclic enkephalins with a diversely substituted guanidine bridge or a thiourea bridge: synthesis, biological and structural evaluations.
University of Montpellier
Synthesis and changes in affinity for NOP and opioid receptors of novel hexapeptides containing β(2)-tryptophan analogues.
Bulgarian Academy of Sciences
Ac-[3- and 4-alkylthioproline31]-CCK4 analogs: synthesis and implications for the CCK-B receptor-bound conformation.
Washington University
Synthesis and biological activity of new peptide segments of gastrin exhibiting gastrin antagonist property.
TBA
Receptor-Ligand Interaction Measured by Inductively Coupled Plasma Mass Spectrometry and Selenium Labeling.
University of Montpellier
Synthesis and biological activity of partially modified retro-inverso pseudopeptide derivatives of the C-terminal tetrapeptide of gastrin.
TBA
Synthesis of gastrin antagonists, analogues of the C-terminal tetrapeptide of gastrin, by introduction of a beta-homo residue.
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues.
University of Montpellier
Synthesis and structure-activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring.
Universit�� Degli Studi Di Parma
Adenosine receptor agonists: synthesis and biological evaluation of the diastereoisomers of 2-(3-hydroxy-3-phenyl-1-propyn-1-yl)NECA.
UniversitÀ