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18 articles for E Altmann


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure-based design and optimization of potent inhibitors of the adenoviral protease.EBI
Novartis Institute For Biomedical Research
Penta-substituted benzimidazoles as potent antagonists of the calcium-sensing receptor (CaSR-antagonists).EBI
Novartis Institutes For Biomedical Research
1-Alkyl-4-phenyl-6-alkoxy-1H-quinazolin-2-ones: a novel series of potent calcium-sensing receptor antagonists.EBI
Novartis Institutes For Biomedical Research
Novel purine nitrile derived inhibitors of the cysteine protease cathepsin K.EBI
Novartis Institutes For Biomedical Research
Arylaminoethyl amides as inhibitors of the cysteine protease cathepsin K-investigating P1' substituents.EBI
Novartis Pharma
Arylaminoethyl amides as novel non-covalent cathepsin K inhibitors.EBI
TBA
Discovery of Potent, Highly Selective, and EBI
Novartis Institutes For Biomedical Research
Structure-Based Design and Preclinical Characterization of Selective and Orally Bioavailable Factor XIa Inhibitors: Demonstrating the Power of an Integrated S1 Protease Family Approach.EBI
Novartis Institutes For Biomedical Research
7-Pyrrolidinyl- and 7-piperidinyl-5-aryl-pyrrolo[2,3-d]pyrimidines--potent inhibitors of the tyrosine kinase c-Src.EBI
Novartis Pharma Research
7-Alkyl- and 7-cycloalkyl-5-aryl-pyrrolo[2,3-d]pyrimidines--potent inhibitors of the tyrosine kinase c-Src.EBI
Novartis Pharma Research
Substituted 5,7-diphenyl-pyrrolo[2,3d]pyrimidines: potent inhibitors of the tyrosine kinase c-Src.EBI
Novartis Pharma
Design, Synthesis, and Experimental Validation of Peptide Ligands Targeting Mycobacterium tuberculosis s Factors.BDB
Indian Institute of Science
Heteroaryloxycarbocyclyl compounds as PDE10 inhibitorsBDB
Amgen
Inhibitors of protein kinasesBDB
Portola Pharmaceuticals
Design and synthesis of paracaseolide A analogues as selective protein tyrosine phosphatase 1B inhibitors.BDB
Lanzhou University
Receptor binding, behavioral, and electrophysiological profiles of nonpeptide corticotropin-releasing factor subtype 1 receptor antagonists CRA1000 and CRA1001.BDB
Taisho Pharmaceutical
Oxindole-based inhibitors of cyclin-dependent kinase 2 (CDK2): design, synthesis, enzymatic activities, and X-ray crystallographic analysis.BDB
Glaxosmithkline
Imidazo[1,2-b]pyridazines: a potent and selective class of cyclin-dependent kinase inhibitors.BDB
Astrazeneca