BDBM7945 1-(trimethylsilyl)-1H-imidazole::Imidazole N-1 deriv. 6::N-(Trimethylsilyl)-imidazole

SMILES C[Si](C)(C)n1ccnc1

InChI Key InChIKey=YKFRUJSEPGHZFJ-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 7945   

TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

LigandPNGBDBM7945(1-(trimethylsilyl)-1H-imidazole | Imidazole N-1 de...)
Affinity DataKi:  1.67E+5nM ΔG°:  -5.24kcal/molepH: 8.0 T: 2°CAssay Description:QC activity was evaluated fluorometrically using Gln-AMC as substrate, and pyroglutamyl peptidase as the auxiliary enzyme. After conversion of Gln-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed