BDBM725057 N-(2-chloro-4-(2- (cyclopropanecarboxamido) pyridin-4-yl)-3- fluorobenzyl)-5-(1- methylcyclopropyl)-1,2,4- oxadiazole-3-carboxamide::US12240838, Compound 59

SMILES CC1(c2nc(C(=O)NCc3ccc(-c4ccnc(NC(=O)C5CC5)c4)c(F)c3Cl)no2)CC1

InChI Key InChIKey=PWFKHIMFQYSXKU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 725057   

TargetTyrosine-protein kinase BTK(Human)
Biogen Ma

US Patent
LigandPNGBDBM725057(N-(2-chloro-4-(2- (cyclopropanecarboxamido) pyridi...)
Affinity DataIC50: 1nMAssay Description:The purpose of the BTK in vitro assay is to determine compound potency against BTK through the measurement of IC50. Compound inhibition is measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/6/2025
Entry Details
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