BDBM50075877 4-[5,5-Dimethyl-8-(5-methyl-thiophen-2-yl)-5,6-dihydro-anthracen-2-yl]-benzoic acid::CHEMBL165417
SMILES Cc1ccc(s1)C1=CCC(C)(C)c2cc3ccc(cc3cc12)-c1ccc(cc1)C(O)=O
InChI Key InChIKey=VGAAIQMKJKFJSO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50075877
Affinity DataKd: 11nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor betaMore data for this Ligand-Target Pair