BDBM50236885 CHEMBL4088788
SMILES [H][C@]12CCC[C@H](N3CC[C@H](O)C3)[C@@]1([H])N(CCN2S(C)(=O)=O)C(=O)Cc1ccc(Cl)c(F)c1
InChI Key InChIKey=CRCNINUFPZHOIF-LDBRAYGESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50236885
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 308nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair