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Found 17 Enz. Inhib. hit(s) with Target = 'Coagulation factor XIII A chain [Q652E]'
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185173(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50:  3.70E+4nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185180([2-[[2-(4-tert-Butoxycarbonylpiperazin-1-yl)-2-oxo...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185155([2-[[2-(4-Benzyloxycarbonylpiperazin-1-yl)-2-oxo-e...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185161(Dimethyl-[2-[[2-[4-(2-naphthylmethoxycarbonyl)pipe...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185162(2-Naphthylmethyl 4-[2-(prop-2-enoylamino)acetyl]pi...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185163((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-[(2-brom...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM60581([2-[[2-[4-[(6-Methoxycarbonyl-2-naphthyl)methoxyca...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185164((6-Methoxycarbonyl-2-naphthyl)methyl 4-[2-(prop-2-...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185168([2-[[2-[4-[(4-Methoxycarbonylphenyl)methoxycarbony...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185170(N-[2-[4-(adamantane-1-carbonyl)piperazin-1-yl]-2-o...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185172([2-[[2-[4-(Adamantane-1-carbonyl)piperazin-1-yl]-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185183(2-(1-Adamantyl)ethyl 4-[2-[(2-bromoacetyl)amino]ac...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185176([2-[[2-[4-(1-Adamantylmethoxycarbonyl)piperazin-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185177(1-Adamantylmethyl 4-[2-(prop-2-enoylamino)acetyl]p...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185179(2-(1-Adamantyl)ethyl 4-[2-(prop-2-enoylamino)acety...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))
Aston University

LigandPNGBDBM185182([2-[[2-[4-[[5-(Dimethylamino)-1-naphthyl]sulfonyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:For measurement of TG2 activity, the incorporation of biotinylated cadaverineinto immobilized N,N-dimethylcasein was used as described previously (Wa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed