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Found 2 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A43'
TargetCytochrome P450 3A43(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50252659((S)-N-(1-(3-bromo-4-(piperidin-4-yloxy)benzyl)pyrr...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A43(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM562067(US11396516, Example 2)
Affinity DataIC50:  9.30E+3nMAssay Description:The ability of the tested compounds to inhibit a panel of CYP enzymes in vitro was assessed using a series of human liver microsome assays. Half-maxi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent