Affinity DataIC50: 0.0240nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against procollagen C-proteinase (PCP).More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against procollagen C-proteinase (PCP).More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against procollagen C-proteinase (PCP).More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against procollagen C-proteinase (PCP).More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human JNK2 alpha2 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human JNK2 alpha2 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against Procollagen C-Proteinase (PCP)More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into myelin basic proteinMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human JNK1 alpha1 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibitory effect against Procollagen C-terminal proteinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human JNK2 alpha2 using GST-tagged ATF2 as substrate and [gamma33P]ATP incubated for 10 mins prior to substrate addition measured after...More data for this Ligand-Target Pair