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Found 131 with Last Name = 'adrian' and Initial = 'fj'
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59116(Hymenialdisine, 27k)
Affinity DataIC50: >10nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59148(Hymenialdisine, 28z)
Affinity DataIC50:  12nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59146(Hymenialdisine, 28w)
Affinity DataIC50:  12nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59137(Hymenialdisine, 28p)
Affinity DataIC50:  32nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  37nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59109(Hymenialdisine, 27a)
Affinity DataIC50:  47nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)
Affinity DataIC50:  47nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59113(Hymenialdisine, 27g)
Affinity DataIC50:  48nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59140(Hymenialdisine, 28ai)
Affinity DataIC50:  50nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59139(Hymenialdisine, 28aa)
Affinity DataIC50:  50nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59108(Hymenialdisine, 27b)
Affinity DataIC50:  51nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM50256043((Z)-3-bromohymenialdisine | CHEMBL480350 | Hymenia...)
Affinity DataIC50:  51nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59107(Hymenialdisine, 27c)
Affinity DataIC50:  52nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM50256043((Z)-3-bromohymenialdisine | CHEMBL480350 | Hymenia...)
Affinity DataIC50:  56nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59142(Hymenialdisine, 28n)
Affinity DataIC50:  59nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)
Affinity DataIC50:  62nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59149(Hymenialdisine, 28v)
Affinity DataIC50:  63nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)
Affinity DataIC50:  64nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  70nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM7491((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  73nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59144(Hymenialdisine, 28ac)
Affinity DataIC50:  75nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59102(Hymenialdisine, 9)
Affinity DataIC50:  79nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59130(Hymenialdisine, 28t)
Affinity DataIC50:  81nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59143(Hymenialdisine, 28ad)
Affinity DataIC50:  81nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59148(Hymenialdisine, 28z)
Affinity DataIC50:  88nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59102(Hymenialdisine, 9)
Affinity DataIC50:  90nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59113(Hymenialdisine, 27g)
Affinity DataIC50:  109nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  111nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  112nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59136(Hymenialdisine, 28ah)
Affinity DataIC50:  118nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59110(Hymenialdisine, 27e)
Affinity DataIC50:  120nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59131(Hymenialdisine, 28g)
Affinity DataIC50:  125nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59139(Hymenialdisine, 28aa)
Affinity DataIC50:  147nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59114(Hymenialdisine, 27i)
Affinity DataIC50:  163nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59130(Hymenialdisine, 28t)
Affinity DataIC50:  171nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59115(Hymenialdisine, 27j)
Affinity DataIC50:  175nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59150(Hymenialdisine, 28ae)
Affinity DataIC50:  177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM50256044(5-(2-amino-4-oxo-1H-imidazol-5(4H)-ylidene)-2,3,4,...)
Affinity DataIC50:  177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59107(Hymenialdisine, 27c)
Affinity DataIC50:  177nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59134(Hymenialdisine, 28ab)
Affinity DataIC50:  179nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59114(Hymenialdisine, 27i)
Affinity DataIC50:  187nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59108(Hymenialdisine, 27b)
Affinity DataIC50:  191nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59109(Hymenialdisine, 27a)
Affinity DataIC50:  213nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59103(Hymenialdisine, 15)
Affinity DataIC50:  220nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM16591((4Z)-4-(2-amino-5-oxo-3,5-dihydro-4H-imidazol-4-yl...)
Affinity DataIC50:  250nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59104(Hymenialdisine, 18)
Affinity DataIC50:  251nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59104(Hymenialdisine, 18)
Affinity DataIC50:  268nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59105(Hymenialdisine, 16)
Affinity DataIC50:  363nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59131(Hymenialdisine, 28g)
Affinity DataIC50:  399nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

LigandPNGBDBM59112(Hymenialdisine, 27h)
Affinity DataIC50:  400nMpH: 7.2Assay Description:In vitro kinase assay using SPA assay kit from Amersham Pharmacia Biotech, Uk.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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