Affinity DataKi: 0.0670nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 0.0970nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.25nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.320nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.330nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.620nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.720nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.800nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 0.950nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 6nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 18nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBP linked to ion channel portion of 5-HT3A receptor expressed in HEK293 cells after 4 hrs b...More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBP linked to ion channel portion of 5-HT3A receptor expressed in HEK293 cells after 4 hrs b...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBP linked to ion channel portion of 5-HT3A receptor expressed in HEK293 cells after 4 hrs b...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 136nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 170nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 190nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 295nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 847nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBP linked to ion channel portion of 5-HT3A receptor expressed in HEK293 cells after 4 hrs b...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 9.97E+3nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinities for alpha 4 beta 2 nAChR were determined in tissue suspension of rat cortical membranes using 1 nM [3H]cytisine. Binding affiniti...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Neurosearch
Curated by PDSP Ki Database
Neurosearch
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: 1.70E+5nMAssay Description:Displacement of [3H]MLA from rat nAChR alpha7 linked to ion channel portion of 5-HT3A receptor expressed in human tsA-201 cells after 2.5 hrs by scin...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Copenhagen
University Of Copenhagen
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]MLA from rat nAChR alpha7 linked to ion channel portion of 5-HT3A receptor expressed in human tsA-201 cells after 2.5 hrs by scin...More data for this Ligand-Target Pair