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Found 40 with Last Name = 'akinaga' and Initial = 's'
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50275347(4-(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-2-(2-(py...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276003(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N4-propyl-N...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50024270(CHEMBL85612)
Affinity DataIC50: <10nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128843(16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricy...)
Affinity DataIC50:  13nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128852(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  14nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128851(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  17nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128859(16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50275348(3-(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-2-(2-(py...)
Affinity DataIC50:  34nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276053(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N4-methyl-N...)
Affinity DataIC50:  35nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128846(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  43nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054109(CHEMBL3319301)
Affinity DataIC50:  44nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276056(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N4-phenyl-N...)
Affinity DataIC50:  47nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128850(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  54nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128847(10-Oxime radicicol | 16-Chloro-17,19-dihydroxy-4-m...)
Affinity DataIC50:  56nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276054(2-(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-2-(2-(py...)
Affinity DataIC50:  63nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128857(16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricy...)
Affinity DataIC50:  67nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128853(16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricy...)
Affinity DataIC50:  70nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50275349(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-ethoxy-N-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50275346(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N2-(2-(pyri...)
Affinity DataIC50:  106nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054192(CHEMBL3319304)
Affinity DataIC50:  110nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054192(CHEMBL3319304)
Affinity DataIC50:  110nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054187(CHEMBL3319303)
Affinity DataIC50:  111nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054187(CHEMBL3319303)
Affinity DataIC50:  111nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054136(CHEMBL3319302)
Affinity DataIC50:  120nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276057(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N2-(2-(pyri...)
Affinity DataIC50:  134nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128845(16-Chloro-17,19-dihydroxy-4-methyl-3,7-dioxa-tricy...)
Affinity DataIC50:  140nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50073099((9E,11E)-(4R,6R,8R)-16-chloro-17,19-dihydroxy-4-me...)
Affinity DataIC50:  180nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128854(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  210nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128842(CHEMBL84714 | [2-(16-Chloro-17,19-dihydroxy-4-meth...)
Affinity DataIC50:  360nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50275746(5-(5-methyl-1,3,4-oxadiazol-2-yl)-N4-propyl-N2-(2-...)
Affinity DataIC50:  373nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128860(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50:  390nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50276055(5-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-N4-(2-(meth...)
Affinity DataIC50:  515nMAssay Description:Inhibition of GST-tagged FLT3 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50054108(CHEMBL3356912)
Affinity DataIC50:  520nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128861(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128863(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128864(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128848(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128844(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rattus norvegicus)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128858(2-(16-Chloro-17,19-dihydroxy-4-methyl-2-oxo-3,7-di...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of v-Src tyrosine kinase autophosphorylation in SR3Y1 cells after 15 hr exposureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Kyowa Hakko Kirin

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed