Compile Data Set for Download or QSAR
maximum 50k data
Found 310 with Last Name = 'albanese' and Initial = 'm'
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325449(1-(2-(piperidin-1-yl)ethyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325450(1-(2-(dimethylamino)ethyl)-3-(1-(1-(pyridin-4-ylme...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325465(1-benzyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-4-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325466(1-(3-(dimethylamino)propyl)-3-(1-(1-(pyridin-4-ylm...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325460(1-(4-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325461(1-(3-methoxybenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pi...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325473(1-isobutyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325448(1-(2-morpholinoethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325469(1-(2-isopropoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325467(1-(3-ethoxypropyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325462(1-(4-chlorobenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325472(1-(2-hydroxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108281(CHEMBL32197 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177543(1-(3-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108271(CHEMBL32124 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108260(1-(5-tert-Butyl-[1,2,4]oxadiazol-3-ylmethoxy)-3-(3...)
Affinity DataKi:  1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325470(1-(2-ethoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pipe...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325451(1-(1-(1-(pyridin-4-ylmethyl)piperidine-4-carbonyl)...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108281(CHEMBL32197 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108267(CHEMBL32537 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108272(CHEMBL33249 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108271(CHEMBL32124 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325463(1-(3-chlorobenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108272(CHEMBL33249 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325471(1-(2-methoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108238(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-5-(4-hydro...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108240(5-Methyl-thiophene-2-carboxylic acid {3-(3,4-dichl...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108242(CHEMBL286646 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hyd...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108256(CHEMBL33243 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325468(1-(2-phenoxyethyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177538(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177536(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177530(4-((1H-imidazol-4-yl)methyl)-1-(3-(3-(cyclohexylox...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108265(CHEMBL36462 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50112009(1-(2,6-Dichloro-pyridin-4-yl)-3-[4-(1H-imidazol-4-...)
Affinity DataKi:  3nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108256(CHEMBL33243 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177531(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177535(CHEMBL379445 | N-(4-(3-(4-((1H-imidazol-4-yl)methy...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50175839(4-((1H-imidazol-4-yl)methyl)-1-(3-phenoxypropyl)pi...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177551(4-((1H-imidazol-4-yl)methyl)-N-(thiazol-2-yl)piper...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50177542(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108248(1-(4-tert-Butyl-benzyloxy)-3-(3,4-dichloro-phenyl)...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108251(CHEMBL32309 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  4nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM86188(CHEMBL366977 | SCH 79687)
Affinity DataKi:  4nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108238(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-5-(4-hydro...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108245(5-Bromo-N-{3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108237(CHEMBL418224 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hyd...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325474(1-methyl-3-(1-(1-(pyridin-4-ylmethyl)piperidine-4-...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50325464(1-(2-chlorobenzyl)-3-(1-(1-(pyridin-4-ylmethyl)pip...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]Nalpha-methylhistamine from histamine H3 receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50112024(1-(3-Cyano-phenyl)-3-[4-(1H-imidazol-4-ylmethyl)-b...)
Affinity DataKi:  5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 310 total ) | Next | Last >>
Jump to: