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Found 24 with Last Name = 'allenby' and Initial = 'g'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334841(CHEMBL1643199 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50:  70nMAssay Description:Induction of PPARdelta-mediated PDK4 mRNA upregulation in human myoblast after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334834(2-(4-((2-(2,4-dichlorophenylcarbamoyl)pyrrolidin-1...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334835(2-(4-((3-(2,4-dichlorophenylcarbamoyl)pyrrolidin-1...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334836(CHEMBL1643194 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334837(2-(4-((1-(2,5-dichlorophenylcarbamoyl)isoindolin-2...)
Affinity DataEC50:  320nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334838(2-(4-((1-(4-chlorophenylcarbamoyl)isoindolin-2-yl)...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334839(2-(2-methyl-4-((1-(phenylcarbamoyl)isoindolin-2-yl...)
Affinity DataEC50: >6.00E+4nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334840(2-(4-(carboxymethoxy)-3-methylbenzyl)isoindoline-1...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334841(CHEMBL1643199 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334842((S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334843((R)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334844(CHEMBL1643202 | rac-2-(4-((6-(2,4-dichlorophenylca...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334845(CHEMBL1643203 | rac-2-(4-((7-(2,4-dichlorophenylca...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334836(CHEMBL1643194 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at GAL4-fused human PPARalpha DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334836(CHEMBL1643194 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at GAL4-fused human PPARgamma DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334841(CHEMBL1643199 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at GAL4-fused human PPARgamma DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334841(CHEMBL1643199 | rac-2-(4-((1-(2,4-dichlorophenylca...)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at GAL4-fused human PPARalpha DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334843((R)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at GAL4-fused human PPARalpha DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334842((S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at GAL4-fused human PPARalpha DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334842((S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at GAL4-fused human PPARgamma DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334843((R)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at GAL4-fused human PPARgamma DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50334842((S)-2-(4-((3-(2,4-dichlorophenylcarbamoyl)-3,4-dih...)
Affinity DataEC50:  15nMAssay Description:Induction of PPARdelta-mediated PDK4 mRNA upregulation in human myoblast after 24 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50312463(2-(4-((cyclohexyl(2-(2,4-dichlorophenylamino)-2-ox...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at GAL4-fused human PPARdelta DNA binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed