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Found 61 with Last Name = 'alsharif' and Initial = 'w'
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536985(CHEMBL4531345)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536979(CHEMBL4542088)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM312202(US9604926, Compound CM-397 | US9724435, Compound C...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353848(CHEMBL1831159)
Affinity DataKi:  2.13nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536983(CHEMBL4537047)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM312201(US9604926, Compound CM-396 | US9724435, Compound C...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353845(CHEMBL1830149 | US9604926, Compound CM-341 | US972...)
Affinity DataKi:  3.28nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.35nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353844(CHEMBL270341 | US9604926, Compound CM-145 | US9724...)
Affinity DataKi:  4.17nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536981(CHEMBL4577544)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536984(CHEMBL4589807)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353859(CHEMBL1831158)
Affinity DataKi:  5.33nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536986(CHEMBL4580186)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353849(CHEMBL1831160)
Affinity DataKi:  14.6nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50035105(1'-{4-[1-(4-fluorophenyl)-1H-3-indolyl]butyl}spiro...)
Affinity DataKi:  17nMAssay Description:Binding affinity to sigma 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM312218(US9604926, Compound CM-728 | US9724435, Compound C...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536980(CHEMBL4573555)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536982(CHEMBL4525954)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353856(CHEMBL1831167)
Affinity DataKi:  34.5nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM312201(US9604926, Compound CM-396 | US9724435, Compound C...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536985(CHEMBL4531345)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353846(CHEMBL1831156 | US9604926, Compound CM-338 | US972...)
Affinity DataKi:  71.5nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536986(CHEMBL4580186)
Affinity DataKi:  72nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat brain membranes after 120 mins in presence of (+)-pentazocine by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353853(CHEMBL1831164 | US9604926, Compound CM-349 | US972...)
Affinity DataKi:  90.9nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353850(CHEMBL1831161)
Affinity DataKi:  92.4nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353847(CHEMBL1831157 | US9604926, Compound CM-360 | US972...)
Affinity DataKi:  141nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM312218(US9604926, Compound CM-728 | US9724435, Compound C...)
Affinity DataKi:  144nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536980(CHEMBL4573555)
Affinity DataKi:  166nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353851(CHEMBL1831162)
Affinity DataKi:  222nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536981(CHEMBL4577544)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536979(CHEMBL4542088)
Affinity DataKi:  273nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353857(CHEMBL1831168)
Affinity DataKi:  279nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353855(CHEMBL1831166 | US9604926, Compound CM-361 | US972...)
Affinity DataKi:  295nMAssay Description:Displacement of [125I]RTI-55 from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536983(CHEMBL4537047)
Affinity DataKi:  299nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM312202(US9604926, Compound CM-397 | US9724435, Compound C...)
Affinity DataKi:  366nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536981(CHEMBL4577544)
Affinity DataKi:  446nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter in rat brainstem membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353855(CHEMBL1831166 | US9604926, Compound CM-361 | US972...)
Affinity DataKi:  544nMAssay Description:Displacement of [3H]YM-09151-2 from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353858(CHEMBL1831169)
Affinity DataKi:  614nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353852(CHEMBL1831163)
Affinity DataKi:  714nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536984(CHEMBL4589807)
Affinity DataKi:  724nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536985(CHEMBL4531345)
Affinity DataKi:  752nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353855(CHEMBL1831166 | US9604926, Compound CM-361 | US972...)
Affinity DataKi:  870nMAssay Description:Displacement of [3H]YM-09151-2 from human D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50536982(CHEMBL4525954)
Affinity DataKi:  988nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536981(CHEMBL4577544)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](-)-sulpiride from dopamine D2 receptor in rat brain membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536981(CHEMBL4577544)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]WIN 35428 from dopamine transporter in rat striatal membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536985(CHEMBL4531345)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]WIN 35428 from dopamine transporter in rat striatal membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50536985(CHEMBL4531345)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter in rat brainstem membranes after 120 mins by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50353854(CHEMBL1831165 | US9604926, Compound CM-350 | US972...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma 1 receptor in rat brain membrane after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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