Affinity DataKi: 140nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human plasma BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of human plasma BuChE using butyrylthiocholine as substrate preincubated for 5 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrate preincubated for 5 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 114nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 118nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 131nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
TargetGlyceraldehyde-3-phosphate dehydrogenase(Oryctolagus cuniculus)
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of rabbit muscle GAPDH assessed as residual enzyme activity after 60 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant BuChE (29 to 602 residues) using butyrylthiocholine iodide as substrate preincubated for 5 min...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 198nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
TargetGlyceraldehyde-3-phosphate dehydrogenase(Oryctolagus cuniculus)
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of rabbit muscle GAPDH assessed as residual enzyme activity after 60 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 232nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 245nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 261nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 275nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 276nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 299nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 301nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 301nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
TargetGlyceraldehyde-3-phosphate dehydrogenase(Oryctolagus cuniculus)
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of rabbit muscle GAPDH assessed as residual enzyme activity after 60 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 429nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant BuChE (29 to 602 residues) using butyrylthiocholine iodide as substrate preincubated for 5 min...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 459nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant BuChE (29 to 602 residues) using butyrylthiocholine iodide as substrate preincubated for 5 min...More data for this Ligand-Target Pair
Affinity DataIC50: 473nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant BuChE (29 to 602 residues) using butyrylthiocholine iodide as substrate preincubated for 5 min...More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of porcine brain tubulin polymerization assessed as decrease in fluorescence intensity measured every 60 sec for 90 mins in presence of GT...More data for this Ligand-Target Pair
Affinity DataIC50: 521nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
Affinity DataIC50: 658nMAssay Description:Inhibition of C-terminal 6His-tagged human recombinant AChE (32 to 614 residues) expressed in HEK293 cells using acetylthiocholine iodide as substrat...More data for this Ligand-Target Pair
TargetGlyceraldehyde-3-phosphate dehydrogenase(Oryctolagus cuniculus)
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of rabbit muscle GAPDH assessed as residual enzyme activity after 60 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of porcine brain tubulin polymerization assessed as decrease in fluorescence intensity measured every 60 sec for 90 mins in presence of GT...More data for this Ligand-Target Pair