Affinity DataKi: 0.0251nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0525nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0575nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0603nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Binding affinity to HSP90 under reducing conditions in presence of TECPMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.0680nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Binding affinity to HSP90 under non-reducing conditions in absence of TECPMore data for this Ligand-Target Pair
Affinity DataKi: 0.0759nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.0940nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0977nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Sorbonne University
Curated by PDSP Ki Database
Sorbonne University
Curated by PDSP Ki Database
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Ability to displace [3H]paroxetine bound to Serotonin transporter receptor in rat forebrainMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards Serotonin transporter was determined in rat forebrain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.132nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.141nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Sorbonne University
Curated by PDSP Ki Database
Sorbonne University
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding affinity at recombinant Hsp90alpha incubated for 16 hrs by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Sorbonne University
Curated by PDSP Ki Database
Sorbonne University
Curated by PDSP Ki Database
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Sorbonne University
Curated by PDSP Ki Database
Sorbonne University
Curated by PDSP Ki Database
Affinity DataKi: 0.224nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Ability to displace [3H]granisetron specifically bound to 5-hydroxytryptamine 3 receptor in rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Inhibition of [3H]granisetron binding to 5-hydroxytryptamine 3 receptor (5-HT 3 receptor) of rat cortex and hippocampus tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.234nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:Displacement of [125I]neurokinin A from human recombinant NK2 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Johann Wolfgang Goethe-UniversitäT
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair