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Found 1406 with Last Name = 'beard' and Initial = 'rl'
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101157(US8524917, 130 | US8524917, 165)
Affinity DataIC50:  0.900nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101041(US8524917, 14)
Affinity DataIC50:  1.20nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101040(US8524917, 13)
Affinity DataIC50:  3nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101044(US8524917, 17)
Affinity DataIC50:  3nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101216(US8524917, 189)
Affinity DataIC50:  3nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50029774(4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-naphthalen-2...)
Affinity DataIC50:  3nMAssay Description:Binding affinity towards retinoic acid receptor alpha was determined using [3H]-ATRA (5 nM) as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50097821(4-{(E)-4-[2-(4-Ethyl-phenyl)-6,6-dimethyl-cyclohex...)
Affinity DataIC50:  3nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101190(US8524917, 163)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101050(US8524917, 23)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101038(US8524917, 11 | US8563594, 169)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101219(US8524917, 192)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101038(US8524917, 11 | US8563594, 169)
Affinity DataIC50:  5nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Allergan

Curated by ChEMBL
LigandPNGBDBM50097823(4-[(E)-4-(6,6-Dimethyl-2-p-tolyl-cyclohex-1-enyl)-...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101118(US8524917, 91)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101121(US8524917, 94)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101039(US8524917, 12 | US8563594, 170)
Affinity DataIC50:  6nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101047(US8524917, 20)
Affinity DataIC50:  6nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101055(US8524917, 28)
Affinity DataIC50:  6nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101039(US8524917, 12 | US8563594, 170)
Affinity DataIC50:  6nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101045(US8524917, 18)
Affinity DataIC50:  6.5nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101056(US8524917, 29)
Affinity DataIC50:  7nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101079(US8524917, 52)
Affinity DataIC50:  7nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101131(US8524917, 104)
Affinity DataIC50:  7nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101220(US8524917, 193)
Affinity DataIC50:  8nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101191(US8524917, 164 | US8524917, 169)
Affinity DataIC50:  9nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101191(US8524917, 164 | US8524917, 169)
Affinity DataIC50:  9nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101197(US8524917, 170)
Affinity DataIC50:  9nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101172(US8524917, 145)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101157(US8524917, 130 | US8524917, 165)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101164(US8524917, 137)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327284(N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)thio]-pheny...)
Affinity DataIC50:  10nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327241(N-[5-chloro-2-(methylsulfinyl)phenyl]-1-benzofuran...)
Affinity DataIC50:  11nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101177(US8524917, 150)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101189(US8524917, 162)
Affinity DataIC50:  12nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101116(US8524917, 89)
Affinity DataIC50:  13nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101149(US8524917, 122)
Affinity DataIC50:  13nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101051(US8524917, 24)
Affinity DataIC50:  14nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101053(US8524917, 26)
Affinity DataIC50:  14nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327214(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-3-(...)
Affinity DataIC50:  14nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101096(US8524917, 69)
Affinity DataIC50:  15nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101221(US8524917, 194)
Affinity DataIC50:  15nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101122(US8524917, 95)
Affinity DataIC50:  15nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327296(N-(2-{[(6-aminopyridin-2-yl)methyl]sulfonyl}-5-chl...)
Affinity DataIC50:  15nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101108(US8524917, 81)
Affinity DataIC50:  16nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327306(N-{5-chloro-2-[(1H-pyrazol-3-ylmethyl)thio]phenyl}...)
Affinity DataIC50:  16nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101074(US8524917, 47)
Affinity DataIC50:  17nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM103621(US8563594, 171)
Affinity DataIC50:  17nMAssay Description:FLIPR assay using S1P3 receptor inhibitor.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101120(US8524917, 93)
Affinity DataIC50:  17nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101084(US8524917, 57)
Affinity DataIC50:  18nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM101037(US8524917, 10 | US8563594, 168)
Affinity DataIC50:  19nMAssay Description:Inhibition assay using sphingosine-1-phosphate receptor 3.More data for this Ligand-Target Pair
In DepthDetails US Patent
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