TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Antagonist activity against human progesterone receptor B (hPR-B) in cotransfected CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Serono Pharmaceutical Research Institute
Curated by ChEMBL
Serono Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Inhibitory activity against Protein-tyrosine phosphatase 1BMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 7.60nMAssay Description:Binding affinity for Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Apparent Ki for rat Lanosterol 14-alpha demethylaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for Cytochrome P450 19A1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetCytochrome P450 11B1, mitochondrial(Homo sapiens (Human))
Syntex Discovery Research
Curated by ChEMBL
Syntex Discovery Research
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for corticoid 11-beta-hydroxylaseMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Serono Pharmaceutical Research Institute
Curated by ChEMBL
Serono Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 18nMpH: 5.5Assay Description:Inhibitory activity against Protein-tyrosine phosphatase 1B at pH 5.5More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duke University
Curated by PDSP Ki Database
Duke University
Curated by PDSP Ki Database
Affinity DataKi: 21nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Antagonist activity against human progesterone receptor B (hPR-B) in cotransfected CV-1 cellsMore data for this Ligand-Target Pair